SCHEMBL11065512

SCHEMBL11065512

CCOC(=O)Cc1c(C(=O)O)c2c(n1C)C(=O)c1ccc(F)cc1CC2

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 5/20 0.40
SRD5A1 P18405 1/20 0.37
L3MBTL1 Q9Y468 2/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
AOC3 Q16853 2/20 0.35
LMNA P02545 1/20 0.35
MAPT P10636 1/20 0.35
TSHR P16473 2/20 0.35
ALDH1A1 P00352 2/20 0.35
MEN1 O00255 1/20 0.35
GABRP O00591 1/20 0.35
GABRD O14764 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2D6 P10635 1/20 0.35
GABRA1 P14867 1/20 0.35
GABRB1 P18505 1/20 0.35
GABRG2 P18507 1/20 0.35
GABRB3 P28472 1/20 0.35
GABRA5 P31644 1/20 0.35
CYP2C19 P33261 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11071003 0.92 MAPK14 (0.42) MAPK14SRD5A1SMN1; SMN2AOC3TSHR
SCHEMBL11068179 0.90 L3MBTL1 (0.45) SRD5A1L3MBTL1SMN1; SMN2AOC3LMNA
SCHEMBL11075121 0.90 AKR1B1 (0.39) MAPK14SRD5A1DHODHAKR1B1
SCHEMBL11065609 0.88 HRH1 (0.39) SRD5A1L3MBTL1SMN1; SMN2LMNAMAPT
SCHEMBL11073141 0.86 AKR1B1 (0.42) L3MBTL1SMN1; SMN2LMNAMAPTALDH1A1
SCHEMBL11068485 0.82 L3MBTL1 (0.42) MAPK14SRD5A1L3MBTL1SMN1; SMN2AOC3
SCHEMBL11066911 0.80 KDM1A (0.41) SRD5A1L3MBTL1SMN1; SMN2LMNAMAPT
SCHEMBL11070255 0.80 AKR1B1 (0.40) SRD5A1L3MBTL1LMNAMAPTMEN1
SCHEMBL11182632 0.80 SMN1; SMN2 (0.35) L3MBTL1SMN1; SMN2LMNAMAPTALDH1A1
SCHEMBL11187765 0.79 L3MBTL1 (0.35) L3MBTL1SMN1; SMN2LMNAMAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4444981-A ANTIINFLAMMATORY, ANALGESICS BEECHAM GROUP LIMITED (GB) 1984-04-24 US disclosed
EP-0024807-B1 BENZOCYCLOHEPTAPYRROLEALKANOIC ACIDS AND THEIR DERIVATIVES, PROCESSES FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM BEECHAM GROUP PLC (GB) 1983-11-02 EP disclosed