SCHEMBL11065640

SCHEMBL11065640

CCOC(CN(C(=O)OCc1ccccc1)c1ccc(Cl)cc1)OCC

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.43
MAPT P10636 1/20 0.43
HPGD P15428 1/20 0.43
POLB P06746 2/20 0.41
RXFP1 Q9HBX9 1/20 0.41
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
FFAR1 O14842 1/20 0.39
L3MBTL1 Q9Y468 3/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
PPARG P37231 3/20 0.38
PPARA Q07869 3/20 0.38
CNR2 P34972 1/20 0.38
MAPK1 P28482 1/20 0.37
TP53 P04637 2/20 0.37
LMNA P02545 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11063095 0.89 ALDH1A1 (0.44) ALDH1A1MAPTHPGDPOLBNPC1
SCHEMBL11062234 0.88 ALDH1A1 (0.43) ALDH1A1MAPTHPGDPOLBNPC1
SCHEMBL11065506 0.87 L3MBTL1 (0.50) ALDH1A1L3MBTL1PPARGPPARALMNA
SCHEMBL8248373 0.87 RNF4 (0.47) ALDH1A1MAPTHPGDNPC1RAB9A
SCHEMBL11073272 0.86 ALDH1A1 (0.43) ALDH1A1POLBNPC1CYP1A2CYP3A4
SCHEMBL11068842 0.81 LTB4R2 (0.41) ALDH1A1MAPTHPGDRAB9AFFAR1
SCHEMBL11062393 0.80 L3MBTL1 (0.43) ALDH1A1MAPTHPGDNPC1RAB9A
SCHEMBL29837176 0.79 ALDH1A1 (0.39) ALDH1A1MAPTHPGDPOLBNPC1
SCHEMBL11071581 0.76 ALDH1A1 (0.47) ALDH1A1MAPTHPGDPOLBNPC1
SCHEMBL6575843 0.75 ALDH1A1 (0.44) ALDH1A1MAPTHPGDPOLBNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4447436-A 1,2,3,4-Tetrahydroisoquinolines 6.10,7,8 dihydroxy substitute-1-methylanilino and use as smooth muscle relaxants FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1984-05-08 US disclosed
US-4220647-A MUSCLE RELAXANTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1980-09-02 US disclosed