SCHEMBL11066529

SCHEMBL11066529

Cc1ccc(C2(C(C)(C)O)CCN(C)CC2)s1

nearest known ligand 0.33

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.33
HCAR3 P49019 1/20 0.32
HCAR2 Q8TDS4 1/20 0.32
SLC6A2 P23975 1/20 0.30
SLC6A4 P31645 1/20 0.30
SLC6A3 Q01959 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5754499 0.75 KMT2A (0.43) SLC6A2SLC6A4SLC6A3
SCHEMBL10640876 0.72 OPRM1 (0.49) CYP1A2SLC6A3
SCHEMBL1152677 0.70 OPRM1 (0.49) SLC6A4
SCHEMBL11072043 0.70 CYP1A2 (0.40) CYP1A2SLC6A4
SCHEMBL5754493 0.69 CHRM1 (0.37)
SCHEMBL10637592 0.68 OPRM1 (0.46) SLC6A2SLC6A4SLC6A3
SCHEMBL10637222 0.68 OPRM1 (0.50) SLC6A2SLC6A4SLC6A3
SCHEMBL11075430 0.68 OPRD1 (0.44) SLC6A4
SCHEMBL10637823 0.67 CYP3A4 (0.35) SLC6A4
SCHEMBL10641018 0.66 POLB (0.42)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4485109-A 4-Aryl-4-piperidinecarbinols E. I. DU PONT DE NEMOURS AND COMPANY (US) 1984-11-27 US disclosed
EP-0094018-A2 4-Aryl-4-piperidinecarbinols E.I. DU PONT DE NEMOURS AND COMPANY (US) 1983-11-16 EP disclosed