SCHEMBL11068110

SCHEMBL11068110

CCOC(=O)CCc1ccc2[nH]c(-c3cccnc3)c(C)c2c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 1/20 0.52
CYP11B2 P19099 1/20 0.52
PDE3B Q13370 1/20 0.48
PDE3A Q14432 1/20 0.48
P2RY12 Q9H244 1/20 0.48
MTNR1A P48039 1/20 0.47
MTNR1B P49286 1/20 0.47
MMP2 P08253 1/20 0.46
MMP13 P45452 1/20 0.46
MMP14 P50281 1/20 0.46
TLR9 Q9NR96 1/20 0.44
TUBB4A P04350 1/20 0.42
TUBB P07437 1/20 0.42
TUBA3C P0DPH7 1/20 0.42
TUBA1B P68363 1/20 0.42
TUBA4A P68366 1/20 0.42
TUBB4B P68371 1/20 0.42
TUBB3 Q13509 1/20 0.42
TUBB2A Q13885 1/20 0.42
TUBB8 Q3ZCM7 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL11075166 0.99 CYP11B1 (0.51) CYP11B1CYP11B2PDE3BPDE3AP2RY12
SCHEMBL11069030 0.87 CYP11B1 (0.56) CYP11B1CYP11B2MTNR1AMTNR1BTLR9
Hydrochloric Acid SCHEMBL11075582 0.86 PDE3B (0.50) PDE3BPDE3AP2RY12MMP2MMP13
Hydrochloric Acid SCHEMBL11007766 0.86 CYP11B1 (0.55) CYP11B1CYP11B2MTNR1AMTNR1BTLR9
SCHEMBL10981215 0.81 CYP11B1 (0.53) CYP11B1CYP11B2MTNR1AMTNR1BTUBB4A
SCHEMBL23704287 0.78 CYP11B1 (0.64) CYP11B1CYP11B2MTNR1AMTNR1BTLR9
SCHEMBL29994013 0.78 CYP11B1 (0.64) CYP11B1CYP11B2MTNR1AMTNR1BTLR9
SCHEMBL5068360 0.78 CYP4F2 (0.56) MMP2MMP13MMP14CYP1A2CYP3A4
SCHEMBL10978524 0.76 CYP11B1 (0.50) CYP11B1CYP11B2MTNR1AMTNR1BTUBB4A
SCHEMBL10376060 0.76 MTNR1A (0.50) MTNR1AMTNR1BMMP2MMP13MMP14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4478842-A THROMBOXANE SYNTHETASE INHIBITORS CIBA-GEIGY CORPORATION (US) 1984-10-23 US disclosed
US-4460777-A THROMBOXANE SYNTHETASE INHIBITORS CIBA-GEIGY CORPORATION (US) 1984-07-17 US disclosed
EP-0080154-A2 N-substituted 2-pyridyl indoles, process for their preparation, pharmaceutical compositions containing them, and their therapeutical use CIBA-GEIGY AG (CH) 1983-06-01 EP disclosed