SCHEMBL11069030

SCHEMBL11069030

Cc1c(-c2cccnc2)[nH]c2ccc(CCC(=O)O)cc12

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 1/20 0.56
CYP11B2 P19099 1/20 0.56
PPARG P37231 5/20 0.55
TBXAS1 P24557 5/20 0.53
MTNR1A P48039 1/20 0.48
MTNR1B P49286 1/20 0.48
TLR9 Q9NR96 1/20 0.46
FFAR1 O14842 6/20 0.44
TUBB4A P04350 1/20 0.43
TUBB P07437 1/20 0.43
TUBA3C P0DPH7 1/20 0.43
TUBA1B P68363 1/20 0.43
TUBA4A P68366 1/20 0.43
TUBB4B P68371 1/20 0.43
TUBB3 Q13509 1/20 0.43
TUBB2A Q13885 1/20 0.43
TUBB8 Q3ZCM7 1/20 0.43
TUBA3E Q6PEY2 1/20 0.43
TUBA1A Q71U36 1/20 0.43
TUBA1C Q9BQE3 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL11007766 0.99 CYP11B1 (0.55) CYP11B1CYP11B2PPARGTBXAS1MTNR1A
SCHEMBL11068110 0.87 CYP11B1 (0.52) CYP11B1CYP11B2PPARGTBXAS1MTNR1A
Hydrochloric Acid SCHEMBL11075166 0.86 CYP11B1 (0.51) CYP11B1CYP11B2PPARGTBXAS1MTNR1A
SCHEMBL11070611 0.86 TBXAS1 (0.63) PPARGTBXAS1TLR9FFAR1
Hydrochloric Acid SCHEMBL11005148 0.85 TBXAS1 (0.61) PPARGTBXAS1TLR9FFAR1
SCHEMBL23704287 0.81 CYP11B1 (0.64) CYP11B1CYP11B2MTNR1AMTNR1BTLR9
SCHEMBL29994013 0.81 CYP11B1 (0.64) CYP11B1CYP11B2MTNR1AMTNR1BTLR9
SCHEMBL11091325 0.77 PPARG (0.52) PPARGTBXAS1MTNR1AMTNR1BFNTA
SCHEMBL29994022 0.75 CYP11B1 (0.47) CYP11B1CYP11B2MTNR1AMTNR1BTLR9
SCHEMBL23704400 0.75 CYP11B1 (0.47) CYP11B1CYP11B2MTNR1AMTNR1BTLR9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4478842-A THROMBOXANE SYNTHETASE INHIBITORS CIBA-GEIGY CORPORATION (US) 1984-10-23 US disclosed
US-4460777-A THROMBOXANE SYNTHETASE INHIBITORS CIBA-GEIGY CORPORATION (US) 1984-07-17 US disclosed
EP-0080154-A2 N-substituted 2-pyridyl indoles, process for their preparation, pharmaceutical compositions containing them, and their therapeutical use CIBA-GEIGY AG (CH) 1983-06-01 EP disclosed