SCHEMBL11069719

SCHEMBL11069719

C=CCn1c(=O)c2[nH]c(C)nc2n(CCC(C)C)c1=O

nearest known ligand 0.56

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PDE2A O00408 2/20 0.54
PDE1A P54750 2/20 0.54
PDE1B Q01064 2/20 0.54
PDE1C Q14123 2/20 0.54
ADORA2B P29275 8/20 0.47
ADORA2A P29274 6/20 0.47
PDE4A P27815 1/20 0.45
PDE4B Q07343 1/20 0.45
PDE4C Q08493 1/20 0.45
PDE4D Q08499 1/20 0.45
ADORA3 P0DMS8 1/20 0.41
ADORA1 P30542 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10857602 0.89 PDE1A (0.66) PDE2APDE1APDE1BPDE1CADORA2B
SCHEMBL9122677 0.88 ADORA2B (0.55) PDE2APDE1APDE1BPDE1CADORA2B
SCHEMBL10856290 0.86 ADORA2B (0.61) ADORA2BADORA2APDE4APDE4BPDE4C
SCHEMBL4953015 0.84 ADORA2B (0.52) PDE2APDE1APDE1BPDE1CADORA2B
SCHEMBL10855008 0.80 ADORA2A (0.49) PDE2APDE1APDE1BPDE1CADORA2B
SCHEMBL2917587 0.76 PDE1A (0.78) PDE2APDE1APDE1BPDE1CADORA2B
SCHEMBL9429916 0.74 PDE2A (0.53) PDE2APDE1APDE1BPDE1CADORA2B
SCHEMBL4621727 0.73 PDE2A (0.51) PDE2APDE1APDE1BPDE1CADORA2B
SCHEMBL10855561 0.73 PDE2A (0.73) PDE2APDE1APDE1BPDE1CADORA2B
SCHEMBL1063544 0.72 SIRT1 (0.68) ADORA2BADORA2AADORA3ADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4469698-A SEDATIVES, TRANQUILIZERS SOCIETE D'ASSISTANCE TECHNIQUE POUR PRODUITS NESTLE S.A. (CH) 1984-09-04 US claimed