SCHEMBL11069998

SCHEMBL11069998

CSCc1cnc2ccccc2c1O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ERN1 O75460 1/20 0.39
KDM4E B2RXH2 2/20 0.39
GPR3 P46089 1/20 0.39
MAPT P10636 3/20 0.37
MEN1 O00255 3/20 0.37
KMT2A Q03164 3/20 0.37
LOXL2 Q9Y4K0 1/20 0.36
ALDH1A1 P00352 2/20 0.35
HPGD P15428 2/20 0.35
GLA P06280 1/20 0.35
GAA P10253 1/20 0.35
HSD17B10 Q99714 1/20 0.35
DUSP10 Q9Y6W6 1/20 0.35
HTT P42858 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C19 P33261 1/20 0.33
HIF1A Q16665 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15045826 0.81 ERN1 (0.46) ERN1KDM4EGPR3MEN1KMT2A
SCHEMBL3396523 0.80 KDM4E (0.45) ERN1KDM4EGPR3MAPTKMT2A
SCHEMBL3394680 0.77 KDM4E (0.42) ERN1KDM4EGPR3KMT2ALOXL2
SCHEMBL28115761 0.77 KDM4E (0.42) ERN1KDM4EGPR3LOXL2ALDH1A1
SCHEMBL11067317 0.76 HTR1A (0.39) KDM4EMAPTMEN1KMT2AALDH1A1
SCHEMBL7850047 0.75 TLR7 (0.43) KDM4EMAPTALDH1A1HPGDGLA
SCHEMBL25946337 0.75 LOXL2 (0.58) KDM4EMAPTMEN1KMT2ALOXL2
SCHEMBL6529277 0.74 TLR7 (0.48) KDM4EMAPTALDH1A1HPGDGLA
SCHEMBL10595445 0.74 PARP1 (0.46) ERN1KDM4EMAPTKMT2AGAA
SCHEMBL11064349 0.74 ERN1 (0.44) ERN1KDM4EGPR3MAPTLOXL2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4447435-A HYPOTENSIVE AGENTS THE BOOTS COMPANY PLC (GB) 1984-05-08 US disclosed
US-4442109-A 3-Methylthiomethyl-and 3-methylsulfinylmethyl-4-quinolinones useful for treating hypertension THE BOOTS COMPANY LIMITED (GB) 1984-04-10 US disclosed