SCHEMBL11070525

SCHEMBL11070525

CCCCN(CCCC)C1(c2ccc(Cl)cc2)CCC(N(C)CC)CC1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 5/20 0.45
SLC6A3 Q01959 5/20 0.45
OPRM1 P35372 2/20 0.38
OPRL1 P41146 2/20 0.38
KCNH2 Q12809 9/20 0.36
SLC6A2 P23975 2/20 0.34
LMNA P02545 3/20 0.33
ALDH1A1 P00352 2/20 0.33
CHRM2 P08172 1/20 0.33
ADRA2A P08913 1/20 0.33
ADRA2B P18089 1/20 0.33
ADRA2C P18825 1/20 0.33
HTR2A P28223 1/20 0.33
OPRK1 P41145 1/20 0.33
HTR2B P41595 1/20 0.33
PTBP1 P26599 1/20 0.33
NOS3 P29474 1/20 0.33
NOS1 P29475 1/20 0.33
NOS2 P35228 1/20 0.33
CYP3A4 P08684 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11078328 0.92 SLC6A4 (0.47) SLC6A4SLC6A3OPRM1OPRL1KCNH2
SCHEMBL11075649 0.88 SLC6A3 (0.50) SLC6A4SLC6A3OPRL1KCNH2SLC6A2
SCHEMBL11070591 0.85 OPRM1 (0.41) OPRM1OPRL1
SCHEMBL11065844 0.84 OPRM1 (0.34) SLC6A4SLC6A3OPRM1OPRL1KCNH2
SCHEMBL11069810 0.83 SLC6A4 (0.41) SLC6A4SLC6A3KCNH2SLC6A2CHRM2
SCHEMBL11076078 0.81 SLC6A4 (0.49) SLC6A4SLC6A3OPRM1OPRL1KCNH2
SCHEMBL11076146 0.80 HTR1D (0.36) OPRM1OPRL1KCNH2LMNAALDH1A1
SCHEMBL11072605 0.79 SLC6A4 (0.41) SLC6A4SLC6A3KCNH2SLC6A2CHRM2
SCHEMBL11079381 0.78 PGR (0.31) OPRM1OPRL1KCNH2LMNAALDH1A1
SCHEMBL11070520 0.78 MDM2 (0.41) SLC6A4SLC6A3OPRM1OPRL1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4447454-A Analgetic compounds, compositions and process of treatment THE UPJOHN COMPANY (US) 1984-05-08 US disclosed
US-4113866-A ANALGETIC COMPOUNDS, COMPOSITIONS AND PROCESS OF TREATMENT THE UPJOHN COMPANY (US) 1978-09-12 US disclosed