SCHEMBL11071495

SCHEMBL11071495

CC(CCc1ccccc1)NCC(O)COc1ccccc1C#N

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.67
KMT2A Q03164 2/20 0.67
ALDH1A1 P00352 1/20 0.67
HTR1A P08908 1/20 0.59
ADRA2A P08913 1/20 0.59
ADRA2B P18089 1/20 0.59
MAOA P21397 1/20 0.59
HTR2B P41595 1/20 0.59
ADRB2 P07550 8/20 0.53
ADRB3 P13945 7/20 0.53
ADRB1 P08588 7/20 0.53
KDM4E B2RXH2 1/20 0.52
CYP1A2 P05177 1/20 0.52
ALOX15 P16050 1/20 0.52
CYP2D6 P10635 2/20 0.51
SLC6A2 P23975 2/20 0.51
SLC6A4 P31645 2/20 0.51
CASR P41180 2/20 0.51
SLC6A3 Q01959 2/20 0.51
KCNH2 Q12809 2/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11751333 0.84 HTR1A (0.65) MEN1KMT2AALDH1A1HTR1AADRA2A
SCHEMBL11200218 0.83 HTR2B (0.70) ALDH1A1HTR1AADRA2AADRA2BMAOA
SCHEMBL11207616 0.81 HTR1A (0.67) MEN1KMT2AALDH1A1HTR1AADRA2A
SCHEMBL11469815 0.81 HTR1A (0.63) MEN1KMT2AALDH1A1HTR1AADRA2A
SCHEMBL11073795 0.81 MEN1 (0.68) MEN1KMT2AALDH1A1ADRB2ADRB3
SCHEMBL11499698 0.80 ALDH1A1 (0.58) MEN1KMT2AALDH1A1HTR1AADRA2A
SCHEMBL11245319 0.80 ALDH1A1 (0.67) MEN1KMT2AALDH1A1HTR1AADRA2A
SCHEMBL11748169 0.79 HTR1A (0.68) MEN1KMT2AALDH1A1HTR1AADRA2A
SCHEMBL11074646 0.79 MEN1 (0.65) MEN1KMT2AALDH1A1HTR2BADRB2
SCHEMBL11079509 0.79 ALDH1A1 (0.65) MEN1KMT2AALDH1A1HTR1AADRA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4450115-A ADRENERGIC BLOCKING AGENTS; HYPOTENSIVE AND CARDIOTONIC AGENTS KYOWA HAKKO KOGYO CO., LTD. (JP) 1984-05-22 US claimed
US-4450115-A ADRENERGIC BLOCKING AGENTS; HYPOTENSIVE AND CARDIOTONIC AGENTS KYOWA HAKKO KOGYO CO., LTD. (JP) 1984-05-22 US disclosed
US-4381398-A Amino-alcohol derivatives KYOWA HAKKO KOGYO CO., LTD. (JP) 1983-04-26 US disclosed