SCHEMBL11073030

SCHEMBL11073030

CCC(=O)c1ccc(OCBr)c(C)c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.49
KMT2A Q03164 1/20 0.49
THRA P10827 1/20 0.48
THRB P10828 1/20 0.48
TAS1R3 Q7RTX0 3/20 0.47
TAS1R1 Q7RTX1 3/20 0.47
KDM4E B2RXH2 2/20 0.47
SMN1; SMN2 Q16637 2/20 0.46
HPGD P15428 2/20 0.46
NPC1 O15118 1/20 0.46
RAB9A P51151 1/20 0.46
MAPT P10636 2/20 0.44
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
ALDH1A1 P00352 2/20 0.42
POLB P06746 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3948073 0.81 MEN1 (0.60) MEN1KMT2ATAS1R3TAS1R1KDM4E
SCHEMBL28012455 0.80 MEN1 (0.46) MEN1KMT2ATHRATHRBTAS1R3
SCHEMBL6812174 0.79 SMN1; SMN2 (0.73) KDM4ESMN1; SMN2HPGDNPC1RAB9A
SCHEMBL6808384 0.79 KMT2A (0.49) MEN1KMT2ATHRATHRBTAS1R3
SCHEMBL8011974 0.78 MAPT (0.55) MEN1KMT2AKDM4ESMN1; SMN2HPGD
SCHEMBL28162947 0.77 PDE4B (0.47) MEN1KMT2ATHRATHRBTAS1R3
SCHEMBL15943001 0.77 THRA (0.61) THRATHRB
SCHEMBL28012472 0.76 MEN1 (0.44) MEN1KMT2ATHRATHRBTAS1R3
SCHEMBL6808423 0.76 SMN1; SMN2 (0.76) MEN1KMT2ATHRBKDM4ESMN1; SMN2
SCHEMBL10799135 0.75 KMT2A (0.51) MEN1KMT2ATHRATHRBKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4450115-A ADRENERGIC BLOCKING AGENTS; HYPOTENSIVE AND CARDIOTONIC AGENTS KYOWA HAKKO KOGYO CO., LTD. (JP) 1984-05-22 US disclosed