SCHEMBL11074465

SCHEMBL11074465

COc1cccc(CC(C#N)(CCC(=O)O)CCC(=O)O)c1

nearest known ligand 0.48

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.48
CTBP2 P56545 1/20 0.47
FFAR1 O14842 2/20 0.46
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
GRM2 Q14416 1/20 0.44
GRM3 Q14832 1/20 0.44
LMNA P02545 1/20 0.43
EPHX2 P34913 2/20 0.43
SLC13A5 Q86YT5 1/20 0.42
RAB9A P51151 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11091483 0.84 FFAR1 (0.47) FFAR1RAB9A
SCHEMBL11099780 0.78 HDAC1 (0.43) CYP1A2MEN1KMT2ALMNA
SCHEMBL11074467 0.76 LMNA (0.46) CYP1A2FFAR1LMNARAB9A
SCHEMBL346302 0.74 FFAR1 (0.65) CYP1A2FFAR1LMNARAB9A
SCHEMBL29824310 0.74 PTGS1 (0.67) CYP1A2CTBP2MEN1KMT2ALMNA
SCHEMBL229067 0.74 PTGS1 (0.67) CYP1A2CTBP2MEN1KMT2ALMNA
Hydrochloric Acid SCHEMBL8693464 0.73 CTBP2 (0.65) CYP1A2CTBP2MEN1KMT2ALMNA
SCHEMBL8218805 0.73 CTBP2 (0.65) CYP1A2CTBP2MEN1KMT2ALMNA
SCHEMBL8953320 0.72 CYP1A2 (0.51) CYP1A2CTBP2MEN1KMT2ASLC13A5
SCHEMBL227654 0.72 CYP1A2 (0.55) CYP1A2CTBP2MEN1KMT2ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4460604-A ANALGESICS, NARCOTIC ANTAGONIST THE UPJOHN COMPANY (US) 1984-07-17 US disclosed
US-4447454-A Analgetic compounds, compositions and process of treatment THE UPJOHN COMPANY (US) 1984-05-08 US disclosed
US-4180584-A ANALGESIC; NARCOTIC ANTAGONIST THE UPJOHN COMPANY (US) 1979-12-25 US disclosed
US-4113866-A ANALGETIC COMPOUNDS, COMPOSITIONS AND PROCESS OF TREATMENT THE UPJOHN COMPANY (US) 1978-09-12 US disclosed
US-4065573-A ANALGESICS THE UPJOHN COMPANY (US) 1977-12-27 US disclosed