SCHEMBL11075293

SCHEMBL11075293

CN1CC(c2cc(Cl)ccc2Cl)CN=C1N

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 2/20 0.36
ADRA1B P35368 2/20 0.36
SRD5A1 P18405 2/20 0.35
KDM4E B2RXH2 1/20 0.33
USP2 O75604 1/20 0.33
ALDH1A1 P00352 1/20 0.33
MAPT P10636 1/20 0.33
HPGD P15428 1/20 0.33
ALOX15 P16050 1/20 0.33
CASP1 P29466 1/20 0.33
CASP7 P55210 1/20 0.33
KMT2A Q03164 1/20 0.33
HSD17B10 Q99714 1/20 0.33
TP53 P04637 1/20 0.33
TSHR P16473 1/20 0.33
SLC6A3 Q01959 2/20 0.33
TAAR1 Q96RJ0 1/20 0.33
CHRM2 P08172 1/20 0.33
ADRA2A P08913 1/20 0.33
DRD2 P14416 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11082401 0.89 DPP4 (0.39) KDM4EUSP2ALDH1A1MAPTHPGD
SCHEMBL11083189 0.82 ADRA1A (0.40) HTR1AADRA1BTP53TAAR1ADRA2A
SCHEMBL11090881 0.79 SRD5A1 (0.53) SRD5A1TSHRTAAR1DRD2ADRA1A
SCHEMBL11078137 0.77 SLC6A2 (0.41) SLC6A3TAAR1DRD2DRD4SLC6A2
SCHEMBL11085800 0.76 SRD5A1 (0.36) SRD5A1
SCHEMBL11082099 0.75 HTR2C (0.38) HTR1ASRD5A1HTR2AHTR2CHRH1
SCHEMBL11287011 0.74 HTR1A (0.37) HTR1AADRA1BKMT2ASLC6A3CHRM2
SCHEMBL11083392 0.71 BRD4 (0.38) SRD5A1
SCHEMBL11084687 0.71 CHRNB2 (0.38) MAPTALOX15CASP1TP53TSHR
SCHEMBL11082926 0.71 ADRA1A (0.40) HTR1AADRA1BALDH1A1KMT2AADRA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0024776-B1 4-PHENYL AND 5-PHENYL-1,4,5,6-TETRAHYDROPYRIMIDINE DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING SAID DERIVATIVES, AND PROCESS FOR PREPARING SAID DERIVATIVES SYNTEX (U.S.A.) INC. (US) 1984-12-27 EP disclosed
EP-0024776-A1 4-Phenyl and 5-phenyl-1,4,5,6-tetrahydropyrimidine derivatives, pharmaceutical compositions containing said derivatives, and process for preparing said derivatives SYNTEX (U.S.A.) INC. (US) 1981-03-11 EP disclosed