SCHEMBL11075865

SCHEMBL11075865

COc1cccc(CC2(N(C)C)CCC(=O)CC2)c1

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CMA1 P23946 1/20 0.46
AOC3 Q16853 1/20 0.44
MEN1 O00255 3/20 0.43
KMT2A Q03164 3/20 0.43
TAAR1 Q96RJ0 3/20 0.42
IDO1 P14902 2/20 0.42
AGXT P21549 2/20 0.42
SIGMAR1 Q99720 2/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
CALM1 P0DP23 1/20 0.40
CAMKK2 Q96RR4 1/20 0.40
HTR1B P28222 1/20 0.40
CHRM2 P08172 1/20 0.40
CHRM1 P11229 1/20 0.40
CHRM3 P20309 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11092391 0.82 ALDH1A1 (0.43) CMA1AOC3MEN1KMT2AIDO1
SCHEMBL11098005 0.82 AKT2 (0.48) CMA1AOC3MEN1KMT2ATAAR1
SCHEMBL13503885 0.81 HRH3 (0.46) AOC3MEN1KMT2ATAAR1IDO1
SCHEMBL206056 0.80 TAAR1 (0.44) AOC3TAAR1SIGMAR1
SCHEMBL3216894 0.80 TAAR1 (0.44) MEN1KMT2ATAAR1IDO1AGXT
SCHEMBL11073700 0.80 CHRM2 (0.46) CMA1AOC3MEN1KMT2ATAAR1
SCHEMBL208815 0.79 OPRM1 (0.58) MEN1KMT2A
SCHEMBL11073936 0.78 KCNH2 (0.46) CMA1MEN1KMT2ATAAR1IDO1
SCHEMBL11080677 0.78 L3MBTL1 (0.52) MEN1KMT2AL3MBTL1
Ethylene SCHEMBL11075789 0.77 CHRM2 (0.43) CMA1AOC3MEN1KMT2ATAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4460604-A ANALGESICS, NARCOTIC ANTAGONIST THE UPJOHN COMPANY (US) 1984-07-17 US claimed
US-4065573-A ANALGESICS THE UPJOHN COMPANY (US) 1977-12-27 US claimed
US-4460604-A ANALGESICS, NARCOTIC ANTAGONIST THE UPJOHN COMPANY (US) 1984-07-17 US disclosed
US-4447454-A Analgetic compounds, compositions and process of treatment THE UPJOHN COMPANY (US) 1984-05-08 US disclosed
US-4180584-A ANALGESIC; NARCOTIC ANTAGONIST THE UPJOHN COMPANY (US) 1979-12-25 US disclosed
US-4113866-A ANALGETIC COMPOUNDS, COMPOSITIONS AND PROCESS OF TREATMENT THE UPJOHN COMPANY (US) 1978-09-12 US disclosed
US-4065573-A ANALGESICS THE UPJOHN COMPANY (US) 1977-12-27 US disclosed