SCHEMBL11077008

SCHEMBL11077008

CN(C)Cc1cc(Cc2cnc(N[N+](=O)[O-])[nH]c2=O)ccn1

nearest known ligand 0.33

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PLA2G7 Q13093 2/20 0.33
ATAD2 Q6PL18 1/20 0.30
CYP1A2 P05177 1/20 0.30
CYP2D6 P10635 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11082533 0.86 DRD2 (0.34) PLA2G7
SCHEMBL10847559 0.86 PLA2G7 (0.35) PLA2G7CYP1A2CYP2D6
SCHEMBL10848628 0.85 PLA2G7 (0.33) PLA2G7
SCHEMBL11182943 0.83 PLA2G7 (0.31) PLA2G7
SCHEMBL7736057 0.82 PLA2G7 (0.50) PLA2G7
SCHEMBL10618958 0.81 PLA2G7 (0.48) PLA2G7
SCHEMBL10851632 0.78 PARP1 (0.31) CYP2D6
SCHEMBL10848262 0.78 ACHE (0.36)
SCHEMBL10376073 0.78 PLA2G7 (0.42) PLA2G7
SCHEMBL7741977 0.77 IDH1 (0.39)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0039989-B1 PYRIMIDONE DERIVATIVES, PROCESSES FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1984-08-29 EP disclosed
US-4388317-A ANTIHISTAMINES SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1983-06-14 US disclosed
EP-0039989-A1 Pyrimidone derivatives, processes for their preparation and pharmaceutical compositions containing them SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1981-11-18 EP disclosed