SCHEMBL11077087

SCHEMBL11077087

CCSc1cc(SCC)cc(C(CN)CNC)c1

nearest known ligand 0.33

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 3/20 0.33
CYP1A2 P05177 1/20 0.31
HIF1A Q16665 1/20 0.31
HSD17B10 Q99714 1/20 0.31
MAOA P21397 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11080698 0.86 SLC6A4 (0.36) SLC6A4MAOA
SCHEMBL11078963 0.83 SLC6A4 (0.42) SLC6A4HIF1AMAOA
SCHEMBL11077824 0.72 SLC6A2 (0.40) SLC6A4
SCHEMBL11083445 0.72 SLC6A2 (0.33) SLC6A4CYP1A2
SCHEMBL11084940 0.72 SLC6A2 (0.33) SLC6A4CYP1A2HIF1AHSD17B10
SCHEMBL11076375 0.71 MAOA (0.40) SLC6A4CYP1A2HIF1AHSD17B10MAOA
SCHEMBL11079915 0.69 SLC6A4 (0.46) SLC6A4CYP1A2HIF1AHSD17B10MAOA
SCHEMBL2866808 0.68 SLC6A4 (0.39) SLC6A4MAOA
SCHEMBL11088866 0.68 PTGS2 (0.38) SLC6A4HSD17B10MAOA
SCHEMBL11083832 0.68 CYP3A4 (0.33) SLC6A4HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0024776-B1 4-PHENYL AND 5-PHENYL-1,4,5,6-TETRAHYDROPYRIMIDINE DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING SAID DERIVATIVES, AND PROCESS FOR PREPARING SAID DERIVATIVES SYNTEX (U.S.A.) INC. (US) 1984-12-27 EP disclosed
US-4322421-A 4-Phenyl-and 5-phenyl-1,4,5,6-tetrahydro-pyrimidine derivatives SYNTEX (U.S.A.) INC. (US) 1982-03-30 US disclosed
US-4261995-A DISORDERS OF CENTRAL NERVOUS SYSTEM AND CARDIOVASCULAR SYSTEM; HYPOTENSIVE SYNTEX (U.S.A.) INC. (US) 1981-04-14 US disclosed
EP-0024776-A1 4-Phenyl and 5-phenyl-1,4,5,6-tetrahydropyrimidine derivatives, pharmaceutical compositions containing said derivatives, and process for preparing said derivatives SYNTEX (U.S.A.) INC. (US) 1981-03-11 EP disclosed