SCHEMBL11077482

SCHEMBL11077482

CC(=O)Oc1c(C(=O)Nc2ccc(N(C)C)cc2)cnc2ccccc12

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 6/20 0.53
HTR2C P28335 1/20 0.50
HTR2B P41595 1/20 0.50
MAOB P27338 1/20 0.49
MAPT P10636 7/20 0.46
ALDH1A1 P00352 6/20 0.46
MAPK1 P28482 3/20 0.46
NPC1 O15118 3/20 0.46
RAB9A P51151 3/20 0.46
SMN1; SMN2 Q16637 3/20 0.46
TP53 P04637 1/20 0.46
HIF1A Q16665 1/20 0.46
PTGDR2 Q9Y5Y4 1/20 0.45
TDP1 Q9NUW8 3/20 0.44
L3MBTL1 Q9Y468 2/20 0.44
LMNA P02545 1/20 0.44
GAA P10253 1/20 0.44
RECQL P46063 1/20 0.44
MCL1 Q07820 1/20 0.44
HSD17B10 Q99714 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11081196 0.86 POLB (0.52) CYP3A4MAOBNPC1LMNAGAA
SCHEMBL11085958 0.85 CYP3A4 (0.54) CYP3A4MAOBMAPTALDH1A1NPC1
Acetic Acid SCHEMBL11077477 0.82 CYP3A4 (0.57) CYP3A4HTR2CHTR2BMAOBMAPT
SCHEMBL11086777 0.81 MEN1 (0.60) MAPTALDH1A1MAPK1NPC1RAB9A
SCHEMBL11082071 0.78 MAPT (0.58) MAPTALDH1A1NPC1RAB9ASMN1; SMN2
SCHEMBL11083167 0.77 RXFP1 (0.53) MAPTSMN1; SMN2TP53HSD17B10RXFP1
SCHEMBL11082254 0.74 MAPT (0.48) CYP3A4MAPTALDH1A1NPC1RAB9A
SCHEMBL11080819 0.74 LMNA (0.47) MAPTALDH1A1NPC1RAB9ASMN1; SMN2
SCHEMBL11075368 0.71 MAPT (0.49) MAOBMAPTALDH1A1NPC1RAB9A
SCHEMBL28817989 0.70 KDM4E (0.50) CYP3A4MAPTALDH1A1SMN1; SMN2TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4450167-A TRANQUILIZERS; PSYCHOLOGICAL DISORDERS ROUSSEL UCLAF (FR) 1984-05-22 US disclosed