SCHEMBL11078413

SCHEMBL11078413

NCC(CN)c1cccc(Br)c1

nearest known ligand 0.52

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 3/20 0.52
TDO2 P48775 1/20 0.52
HTR2A P28223 3/20 0.45
TAAR1 Q96RJ0 2/20 0.45
C1S P09871 1/20 0.41
AGXT P21549 2/20 0.39
MGAM O43451 1/20 0.39
GAA P10253 1/20 0.39
SI P14410 1/20 0.39
MGAM2 Q2M2H8 1/20 0.39
GABBR2 O75899 1/20 0.38
GABBR1 Q9UBS5 1/20 0.38
ALDH1A1 P00352 1/20 0.38
MAPK1 P28482 1/20 0.38
MAOA P21397 1/20 0.38
HTR2C P28335 1/20 0.37
HTR2B P41595 1/20 0.37
PARP1 P09874 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5775168 0.88 IDO1 (0.42) IDO1TDO2HTR2ATAAR1C1S
SCHEMBL26922035 0.84 HTR2A (0.41) IDO1TDO2HTR2ATAAR1AGXT
SCHEMBL26922629 0.84 HTR2A (0.41) IDO1TDO2HTR2ATAAR1AGXT
SCHEMBL11084001 0.84 SLC6A2 (0.47) IDO1TDO2HTR2ATAAR1GAA
SCHEMBL21610485 0.82 GABBR2 (0.67) GAAGABBR2GABBR1
SCHEMBL23750202 0.81 GABBR2 (0.47) IDO1TDO2MGAMGAASI
Hydrochloric Acid SCHEMBL21609298 0.81 GABBR2 (0.65) IDO1TDO2GAAGABBR2GABBR1
Hydrochloric Acid SCHEMBL29847994 0.81 GABBR2 (0.65) IDO1TDO2GAAGABBR2GABBR1
SCHEMBL4702287 0.81 IDO1 (0.46) IDO1TDO2HTR2ATAAR1AGXT
SCHEMBL1470710 0.81 IDO1 (0.46) IDO1TDO2HTR2ATAAR1AGXT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0024776-B1 4-PHENYL AND 5-PHENYL-1,4,5,6-TETRAHYDROPYRIMIDINE DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING SAID DERIVATIVES, AND PROCESS FOR PREPARING SAID DERIVATIVES SYNTEX (U.S.A.) INC. (US) 1984-12-27 EP disclosed
US-4322421-A 4-Phenyl-and 5-phenyl-1,4,5,6-tetrahydro-pyrimidine derivatives SYNTEX (U.S.A.) INC. (US) 1982-03-30 US disclosed
US-4261995-A DISORDERS OF CENTRAL NERVOUS SYSTEM AND CARDIOVASCULAR SYSTEM; HYPOTENSIVE SYNTEX (U.S.A.) INC. (US) 1981-04-14 US disclosed
EP-0024776-A1 4-Phenyl and 5-phenyl-1,4,5,6-tetrahydropyrimidine derivatives, pharmaceutical compositions containing said derivatives, and process for preparing said derivatives SYNTEX (U.S.A.) INC. (US) 1981-03-11 EP disclosed