SCHEMBL11079784

SCHEMBL11079784

CCc1ccc(C(CC(N)=O)CC(N)=O)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.45
SMN1; SMN2 Q16637 2/20 0.42
TSHR P16473 1/20 0.42
MAPK1 P28482 1/20 0.42
ATM Q13315 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
PLAU P00749 1/20 0.41
EPHX1 P07099 1/20 0.41
F2 P00734 1/20 0.40
F10 P00742 1/20 0.40
IDO1 P14902 2/20 0.40
AKR1C3 P42330 1/20 0.40
AKR1C2 P52895 1/20 0.40
PLK1 P53350 1/20 0.40
LMNA P02545 1/20 0.40
HPGD P15428 1/20 0.40
ESR1 P03372 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2226824 0.82 FFAR1 (0.51) ALDH1A1TSHRMAPK1ATMTDP1
SCHEMBL11075911 0.80 CYP2C19 (0.54) ALDH1A1SMN1; SMN2CYP2C19LMNACYP1A2
SCHEMBL11080642 0.80 ALDH1A1 (0.47) ALDH1A1SMN1; SMN2TSHRMAPK1CYP2C9
SCHEMBL11077922 0.79 ALDH1A1 (0.44) ALDH1A1SMN1; SMN2TSHRMAPK1TDP1
SCHEMBL11073397 0.77 GAA (0.47) ALDH1A1CA2
SCHEMBL11080051 0.77 PARP10 (0.56) ALDH1A1TSHRTDP1AKR1C3AKR1C2
SCHEMBL11080152 0.77 ALDH1A1 (0.42) ALDH1A1SMN1; SMN2
SCHEMBL523877 0.76 GABBR2 (0.59) SMN1; SMN2TSHRCYP2C9CYP2C19LMNA
SCHEMBL11085363 0.76 GABBR2 (0.49) ALDH1A1
SCHEMBL11084494 0.76 ALOX5 (0.46) ALDH1A1SMN1; SMN2EPHX1CA2CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0024776-B1 4-PHENYL AND 5-PHENYL-1,4,5,6-TETRAHYDROPYRIMIDINE DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING SAID DERIVATIVES, AND PROCESS FOR PREPARING SAID DERIVATIVES SYNTEX (U.S.A.) INC. (US) 1984-12-27 EP disclosed
US-4322421-A 4-Phenyl-and 5-phenyl-1,4,5,6-tetrahydro-pyrimidine derivatives SYNTEX (U.S.A.) INC. (US) 1982-03-30 US disclosed
US-4261995-A DISORDERS OF CENTRAL NERVOUS SYSTEM AND CARDIOVASCULAR SYSTEM; HYPOTENSIVE SYNTEX (U.S.A.) INC. (US) 1981-04-14 US disclosed
EP-0024776-A1 4-Phenyl and 5-phenyl-1,4,5,6-tetrahydropyrimidine derivatives, pharmaceutical compositions containing said derivatives, and process for preparing said derivatives SYNTEX (U.S.A.) INC. (US) 1981-03-11 EP disclosed