SCHEMBL11079836

SCHEMBL11079836

CCOC(=O)C(C#N)c1ccsc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.49
MEN1 O00255 2/20 0.49
GAA P10253 2/20 0.49
KMT2A Q03164 2/20 0.49
ALOX5 P09917 1/20 0.41
CHRNB2 P17787 1/20 0.41
CHRNB4 P30926 1/20 0.41
CHRNA3 P32297 1/20 0.41
CHRNA4 P43681 1/20 0.41
MAPT P10636 4/20 0.39
HSD17B10 Q99714 3/20 0.39
ALDH1A1 P00352 3/20 0.39
TSHR P16473 2/20 0.39
CYP1A2 P05177 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
POLB P06746 2/20 0.38
ALOX12 P18054 1/20 0.38
ADORA2B P29275 4/20 0.37
KDM4E B2RXH2 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11384344 0.84 ALOX5 (0.43) SMN1; SMN2MEN1KMT2AALOX5CHRNB2
SCHEMBL17466005 0.82 MEN1 (0.58) SMN1; SMN2MEN1GAAKMT2AMAPT
SCHEMBL8178062 0.79 CHRNB2 (0.46) SMN1; SMN2MEN1GAAKMT2AALOX5
SCHEMBL18734631 0.79 CHRNB2 (0.46) MEN1GAAKMT2AALOX5CHRNB2
SCHEMBL502194 0.78 SMN1; SMN2 (0.61) SMN1; SMN2MEN1GAAKMT2AALDH1A1
SCHEMBL6289274 0.78 SMN1; SMN2 (0.54) SMN1; SMN2MEN1GAAKMT2AALOX5
SCHEMBL10762809 0.78 ALOX5 (0.45) MEN1GAAKMT2AALOX5CHRNB2
SCHEMBL6384665 0.78 ALOX5 (0.45) SMN1; SMN2MEN1GAAKMT2AALOX5
SCHEMBL10772715 0.77 ALOX5 (0.44) SMN1; SMN2ALOX5CHRNB2CHRNB4CHRNA3
SCHEMBL4013434 0.76 CHRNB2 (0.43) MEN1GAAKMT2AALOX5CHRNB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0002846-B1 3-THIENYLMALONIC ACIDS, THE CORRESPONDING DIESTERS AND THEIR PREPARATION Océ-Andeno B.V. (NL) 1984-05-23 EP disclosed
US-4262129-A Preparation of a 3-thienylmalonic acid and the corresponding diesters OCE-ANDENO B.V. (NL) 1981-04-14 US disclosed
US-4252976-A Process for the preparation of thiophenes BEECHAM GROUP LIMITED (DE) 1981-02-24 US disclosed
EP-0002846-A1 3-Thienylmalonic acids, the corresponding diesters and their preparation Océ-Andeno B.V. (NL) 1979-07-11 EP disclosed