SCHEMBL11080503

SCHEMBL11080503

CC(N)C(N)c1cccc(Br)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 1/20 0.46
TDO2 P48775 1/20 0.46
MAOA P21397 1/20 0.44
ALDH1A1 P00352 3/20 0.41
MAPK1 P28482 1/20 0.41
ADRB1 P08588 1/20 0.40
MIF P14174 1/20 0.40
HTR2A P28223 1/20 0.40
ADRA1A P35348 1/20 0.40
HTR2B P41595 1/20 0.40
MBTD1 Q05BQ5 1/20 0.40
L3MBTL3 Q96JM7 1/20 0.40
GBA1 P04062 1/20 0.38
ADRA2A P08913 1/20 0.38
ADRA2C P18825 1/20 0.38
LMNA P02545 1/20 0.38
HIF1A Q16665 1/20 0.38
KDM4E B2RXH2 1/20 0.38
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2401036 0.88 IDO1 (0.46) IDO1TDO2MAOAALDH1A1MAPK1
SCHEMBL29278100 0.88 IDO1 (0.46) IDO1TDO2MAOAALDH1A1MAPK1
SCHEMBL30762162 0.88 IDO1 (0.46) IDO1TDO2MAOAALDH1A1MAPK1
SCHEMBL5772657 0.87 IDO1 (0.52) IDO1TDO2MAOAALDH1A1MAPK1
Hydrochloric Acid SCHEMBL17764461 0.86 IDO1 (0.49) IDO1TDO2MAOAALDH1A1MAPK1
Hydrochloric Acid SCHEMBL30762179 0.86 IDO1 (0.49) IDO1TDO2MAOAALDH1A1MAPK1
SCHEMBL14014456 0.83 IDO1 (0.48) IDO1TDO2MAOAALDH1A1MAPK1
SCHEMBL842088 0.83 IDO1 (0.48) IDO1TDO2MAOAALDH1A1MAPK1
SCHEMBL3689883 0.83 IDO1 (0.48) IDO1TDO2MAOAALDH1A1MAPK1
SCHEMBL749481 0.83 IDO1 (0.48) IDO1TDO2MAOAALDH1A1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108250058-B PPAR agonists and their use in the treatment of Alzheimer's disease and other diseases 上海怡立舍生物技术有限公司 2022-02-11 CN disclosed
EP-0024776-B1 4-PHENYL AND 5-PHENYL-1,4,5,6-TETRAHYDROPYRIMIDINE DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING SAID DERIVATIVES, AND PROCESS FOR PREPARING SAID DERIVATIVES SYNTEX (U.S.A.) INC. (US) 1984-12-27 EP disclosed
US-4322421-A 4-Phenyl-and 5-phenyl-1,4,5,6-tetrahydro-pyrimidine derivatives SYNTEX (U.S.A.) INC. (US) 1982-03-30 US disclosed
US-4261995-A DISORDERS OF CENTRAL NERVOUS SYSTEM AND CARDIOVASCULAR SYSTEM; HYPOTENSIVE SYNTEX (U.S.A.) INC. (US) 1981-04-14 US disclosed
EP-0024776-A1 4-Phenyl and 5-phenyl-1,4,5,6-tetrahydropyrimidine derivatives, pharmaceutical compositions containing said derivatives, and process for preparing said derivatives SYNTEX (U.S.A.) INC. (US) 1981-03-11 EP disclosed