SCHEMBL11080868

SCHEMBL11080868

CCOC(=O)Nc1ccc2c(c1)C(c1ccccc1Cl)SCCC(=O)N2

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.50
TSHR P16473 3/20 0.50
CYP1A2 P05177 3/20 0.50
CYP2C9 P11712 3/20 0.50
CYP2C19 P33261 3/20 0.50
ALOX15 P16050 2/20 0.50
TP53 P04637 1/20 0.50
CASP1 P29466 1/20 0.50
RECQL P46063 1/20 0.50
SLC8B1 Q6J4K2 1/20 0.50
ALDH1A1 P00352 4/20 0.44
LMNA P02545 3/20 0.44
HSD17B10 Q99714 3/20 0.44
KMT2A Q03164 3/20 0.44
MEN1 O00255 2/20 0.44
GAA P10253 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
NOX1 Q9Y5S8 1/20 0.44
DGAT1 O75907 1/20 0.40
POLB P06746 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11087922 0.81 TSHR (0.41) MAPTTSHRCYP1A2CYP2C9CYP2C19
SCHEMBL10929981 0.77 MAPT (0.77) MAPTTSHRCYP1A2CYP2C9CYP2C19
SCHEMBL10929004 0.72 MAPT (0.56) MAPTTSHRCYP1A2CYP2C9CYP2C19
SCHEMBL10367113 0.71 HDAC3 (0.57) MAPTTSHRCYP1A2CYP2C9CYP2C19
SCHEMBL11081504 0.70 ALDH1A1 (0.44) MAPTTSHRCYP1A2CYP2C9CYP2C19
SCHEMBL31071906 0.68 TP53 (1.00) MAPTTSHRCYP1A2CYP2C9CYP2C19
SCHEMBL869274 0.68 TP53 (1.00) MAPTTSHRCYP1A2CYP2C9CYP2C19
SCHEMBL10926019 0.67 MAPT (0.60) MAPTTSHRCYP1A2CYP2C9CYP2C19
SCHEMBL6364379 0.65 KMT2A (0.46) MAPTTSHRCYP1A2CYP2C9CYP2C19
SCHEMBL9659046 0.64 KMT2A (0.70) MAPTTSHRCYP1A2CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4464300-A PSYCHOTROPIC, ANXIOLYTIC AGENTS HOFFMANN-LA ROCHE INC. (US) 1984-08-07 US disclosed