SCHEMBL11081584

SCHEMBL11081584

COc1ccc(/C=C2/CCn3c2nc2ccc(Cl)cc2c3=O)c(OC)c1OC

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 2/20 0.57
NPC1 O15118 1/20 0.57
ALOX5 P09917 2/20 0.54
KMT2A Q03164 6/20 0.52
MEN1 O00255 5/20 0.52
MAPT P10636 2/20 0.52
KDM4E B2RXH2 1/20 0.52
POLB P06746 3/20 0.50
ALDH1A1 P00352 2/20 0.50
THRB P10828 1/20 0.50
HPGD P15428 1/20 0.50
TDP1 Q9NUW8 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.50
TUBB4A P04350 2/20 0.49
TUBB P07437 2/20 0.49
TUBA3C P0DPH7 2/20 0.49
TUBA1B P68363 2/20 0.49
TUBA4A P68366 2/20 0.49
TUBB4B P68371 2/20 0.49
TUBB3 Q13509 2/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11081588 1.00 RAB9A (0.57) RAB9ANPC1ALOX5KMT2AMEN1
SCHEMBL11090606 0.92 RAB9A (0.56) RAB9ANPC1ALOX5KMT2AMEN1
SCHEMBL11090611 0.92 RAB9A (0.56) RAB9ANPC1ALOX5KMT2AMEN1
SCHEMBL11112929 0.88 ALOX5 (0.65) RAB9ANPC1ALOX5KMT2AMEN1
SCHEMBL11112931 0.88 ALOX5 (0.65) RAB9ANPC1ALOX5KMT2AMEN1
SCHEMBL11080914 0.88 RAB9A (0.59) RAB9ANPC1ALOX5KMT2AMEN1
SCHEMBL11080917 0.88 RAB9A (0.59) RAB9ANPC1ALOX5KMT2AMEN1
SCHEMBL11088813 0.87 RAB9A (0.56) RAB9ANPC1ALOX5KMT2AMEN1
SCHEMBL11088808 0.87 RAB9A (0.56) RAB9ANPC1ALOX5KMT2AMEN1
SCHEMBL11087084 0.87 RAB9A (0.61) RAB9ANPC1ALOX5KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4428952-A Substituted pyrrolo[2,1-b]quinazolines and pyrido[2,1-b]quinazolines useful for the treatment of or the prevention of gastrointestinal ulcers FARMITALIA CARLO ERBA S.P.A. (IT) 1984-01-31 US disclosed