SCHEMBL11085254

SCHEMBL11085254

O=C1C2CC2(c2ccccc2)C(=O)N1CCCC(c1ccc(F)cc1)c1ccc(F)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 12/20 0.51
HTR2A P28223 5/20 0.42
ADRA1A P35348 4/20 0.42
HRH1 P35367 4/20 0.42
OPRM1 P35372 4/20 0.42
DRD3 P35462 4/20 0.42
OPRD1 P41143 4/20 0.42
OPRK1 P41145 4/20 0.42
HTR6 P50406 4/20 0.42
SLC6A3 Q01959 4/20 0.42
CACNA1C Q13936 4/20 0.42
HTR2C P28335 3/20 0.42
DRD2 P14416 3/20 0.42
CYP3A4 P08684 3/20 0.42
ADORA3 P0DMS8 3/20 0.42
CYP2D6 P10635 3/20 0.42
MAPK1 P28482 3/20 0.42
MTOR P42345 3/20 0.42
RAB9A P51151 3/20 0.42
MEN1 O00255 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11074234 0.90 CYP19A1 (0.51) CYP19A1DRD3DRD2MEN1LMNA
SCHEMBL8969269 0.75 CYP19A1 (0.62) CYP19A1MAPK1MEN1USP2MAPT
SCHEMBL7430028 0.72 ALDH1A1 (0.64) CYP2D6RAB9ACYP1A2MAPTCYP2C19
SCHEMBL8968925 0.72 CYP19A1 (0.82) CYP19A1MEN1KMT2ASMN1; SMN2TSHR
SCHEMBL11081758 0.70 CYP19A1 (0.76) CYP19A1LMNACYP1A2GAACYP2C9
SCHEMBL6002297 0.69 CYP19A1 (0.72) CYP19A1CYP3A4NPSR1GAAALDH1A1
SCHEMBL11078445 0.68 CYP19A1 (0.71) CYP19A1CYP2C19SMN1; SMN2TSHRALDH1A1
SCHEMBL10529975 0.68 CYP19A1 (1.00) CYP19A1
Fumaric Acid SCHEMBL11077742 0.68 DRD3 (0.45) HTR2AADRA1AHRH1OPRM1DRD3
Fumaric Acid SCHEMBL11077747 0.68 DRD3 (0.45) HTR2AADRA1AHRH1OPRM1DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4435419-A Method of treating depression using azabicyclohexanes AMERICAN CYANAMID COMPANY (US) 1984-03-06 US disclosed
US-4231935-A ANXIOLYTICS AND ANALGESICS AMERICAN CYANAMID COMPANY (US) 1980-11-04 US disclosed
US-4196120-A 1,2-BIS(HYDROCARBYLSULFONYLOXY OR HALO METHYL)CYCLOPROPYLBENZENE, OPTICAL ACITIVITY ANALGESICS AMERICAN CYANAMID COMPANY (US) 1980-04-01 US disclosed
US-4131611-A ANXIOLYTIC, ANALGESIC AMERICAN CYANAMID COMPANY (US) 1978-12-26 US disclosed