SCHEMBL11086602

SCHEMBL11086602

O=C(O)c1cnc2ccsc2c1NNc1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.41
GAA P10253 1/20 0.41
KDR P35968 3/20 0.41
CYP1A2 P05177 1/20 0.41
AURKA O14965 2/20 0.40
PIM1 P11309 1/20 0.40
CDK2 P24941 1/20 0.40
GSK3B P49841 1/20 0.40
AURKB Q96GD4 1/20 0.39
HCRTR1 O43613 1/20 0.37
MAPT P10636 1/20 0.37
ALOX15 P16050 1/20 0.37
TSHR P16473 1/20 0.37
MAPK1 P28482 1/20 0.37
RAB9A P51151 1/20 0.37
HSD17B10 Q99714 1/20 0.37
CSNK2A1 P68400 1/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
EGFR P00533 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11084724 0.88 ALDH1A1 (0.45) ALDH1A1GAACYP1A2AURKAMAPT
SCHEMBL11084270 0.88 MEN1 (0.37) ALDH1A1KDRMAPTMAPK1RAB9A
SCHEMBL11080774 0.85 NPC1 (0.42) ALDH1A1GAAMAPTRAB9AMEN1
SCHEMBL11084914 0.85 KDR (0.46) ALDH1A1GAAKDRMAPTTSHR
SCHEMBL11083402 0.85 CSNK2A1 (0.42) ALDH1A1GAAKDRAURKAAURKB
SCHEMBL11092605 0.85 L3MBTL1 (0.43) GAAKDRCYP1A2PIM1AURKB
SCHEMBL11085398 0.84 MAPT (0.41) ALDH1A1GAAKDRAURKAPIM1
SCHEMBL27301289 0.79 PDE4A (0.53) ALDH1A1MAPTADORA2AADORA2B
SCHEMBL11087340 0.78 SMN1; SMN2 (0.40) ALDH1A1GAAMAPTMAPK1RAB9A
SCHEMBL27297878 0.77 CSNK2A1 (0.47) CSNK2A1MEN1KMT2ACSF1R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0126970-A2 Anxiolytic and anti-depressant thienopyridine derivatives BEECHAM GROUP PLC (GB) 1984-12-05 EP claimed
EP-0126970-A2 Anxiolytic and anti-depressant thienopyridine derivatives BEECHAM GROUP PLC (GB) 1984-12-05 EP disclosed