SCHEMBL11093024

SCHEMBL11093024

COc1ccc2[nH]c(C)c(CC(=O)Oc3ccc(C(=O)OCCN4CCN(C(C)N5CCOCC5)CC4)cc3)c2c1

nearest known ligand 0.50

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 1/20 0.48
ALDH1A1 P00352 7/20 0.46
KDM4E B2RXH2 6/20 0.45
HPGD P15428 2/20 0.45
AKR1C2 P52895 1/20 0.44
SMN1; SMN2 Q16637 2/20 0.42
CYP1A2 P05177 1/20 0.41
HSD17B10 Q99714 3/20 0.41
ALOX15 P16050 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
ATM Q13315 1/20 0.40
KDR P35968 1/20 0.40
GAA P10253 1/20 0.40
LMNA P02545 1/20 0.40
MTNR1A P48039 1/20 0.39
MTNR1B P49286 1/20 0.39
MAPT P10636 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11087764 0.93 PTGS2 (0.54) PTGS2ALDH1A1KDM4EHPGDAKR1C2
Hydrochloric Acid SCHEMBL11093044 0.92 PTGS2 (0.53) PTGS2ALDH1A1KDM4EHPGDAKR1C2
SCHEMBL11192813 0.92 PTGS2 (0.55) PTGS2ALDH1A1KDM4EHPGDAKR1C2
Hydrochloric Acid SCHEMBL11223300 0.92 PTGS2 (0.54) PTGS2ALDH1A1KDM4EHPGDAKR1C2
SCHEMBL11089661 0.88 ALDH1A1 (0.49) PTGS2ALDH1A1KDM4EHPGDAKR1C2
Hydrochloric Acid SCHEMBL11081771 0.87 ALDH1A1 (0.49) PTGS2ALDH1A1KDM4EHPGDAKR1C2
SCHEMBL11093304 0.87 AKR1C2 (0.51) PTGS2ALDH1A1KDM4EHPGDAKR1C2
Hydrochloric Acid SCHEMBL11089910 0.87 AKR1C2 (0.50) PTGS2ALDH1A1KDM4EHPGDAKR1C2
SCHEMBL11197586 0.86 HSD17B10 (0.55) PTGS2ALDH1A1KDM4EHPGDAKR1C2
SCHEMBL11087847 0.83 AKR1C2 (0.46) PTGS2ALDH1A1KDM4EHPGDAKR1C2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4443603-A PROTEOLYTIC ENZYME INHIBITORS KOWA COMPANY LIMITED (JP) 1984-04-17 US disclosed