SCHEMBL11094653

SCHEMBL11094653

CC(CCCN1C(=O)c2ccccc2C1=O)C(=O)CBr

nearest known ligand 0.48

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MAOB P27338 4/20 0.47
ACHE P22303 1/20 0.47
HDAC1 Q13547 5/20 0.46
HDAC7 Q8WUI4 5/20 0.46
HDAC8 Q9BY41 3/20 0.46
HDAC3 O15379 2/20 0.46
HDAC4 P56524 2/20 0.46
HDAC2 Q92769 2/20 0.46
HDAC10 Q969S8 2/20 0.46
HDAC11 Q96DB2 2/20 0.46
HDAC6 Q9UBN7 2/20 0.46
HDAC9 Q9UKV0 2/20 0.46
HDAC5 Q9UQL6 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11093898 0.84 HDAC1 (0.52) MAOBACHEHDAC1HDAC7
SCHEMBL4405142 0.82 ALDH1A1 (0.54)
SCHEMBL11093086 0.81 MAOB (0.45) MAOBHDAC1HDAC7HDAC8HDAC3
SCHEMBL11481918 0.79 HDAC1 (0.58) MAOBACHEHDAC1HDAC7HDAC8
SCHEMBL902525 0.79 MAOB (0.54) MAOB
SCHEMBL28375145 0.79 CHRM2 (0.57) MAOB
SCHEMBL29740550 0.79 CHRM2 (0.57) MAOB
SCHEMBL20472107 0.79 CHRM2 (0.57) MAOB
SCHEMBL1787317 0.78 MAOB (0.56) MAOB
SCHEMBL7438587 0.77 NPC1 (0.50) HDAC1HDAC7HDAC8HDAC3HDAC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0010893-B1 ANTISECRETORY BRANCHED-CHAIN HETEROCYCLIC GUANIDINE DERIVATIVES, PROCESSES FOR THEIR MANUFACTURE, INTERMEDIATES, AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAID DERIVATIVES IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1984-02-08 EP disclosed
EP-0010893-A1 Antisecretory branched-chain heterocyclic guanidine derivatives, processes for their manufacture, intermediates, and pharmaceutical compositions containing said derivatives IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1980-05-14 EP disclosed