SCHEMBL11095028

SCHEMBL11095028

CC(CCCN1C(=O)c2ccccc2C1=O)CC(=O)OCc1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 2/20 0.49
CYP3A4 P08684 1/20 0.49
CYP2D6 P10635 1/20 0.49
CYP2C9 P11712 1/20 0.49
CYP2C19 P33261 1/20 0.49
TDP1 Q9NUW8 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
MAOB P27338 3/20 0.44
CDC25B P30305 1/20 0.44
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
HSD17B10 Q99714 1/20 0.44
MAPK1 P28482 1/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
HDAC1 Q13547 3/20 0.43
HDAC7 Q8WUI4 3/20 0.43
ALDH1A1 P00352 1/20 0.43
SLC15A1 P46059 1/20 0.43
CASP3 P42574 1/20 0.43
MAPT P10636 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11097234 0.82 HDAC1 (0.50) RAB9ATDP1L3MBTL1MAOBMEN1
SCHEMBL6578347 0.81 TDP1 (0.51) RAB9ATDP1L3MBTL1MAOBMAPK1
SCHEMBL6789754 0.80 ALDH1A1 (0.57) TDP1L3MBTL1MEN1KMT2AHSD17B10
SCHEMBL408911 0.79 TDP1 (0.49) RAB9ACYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL10725421 0.79 L3MBTL1 (0.59) TDP1L3MBTL1SMN1; SMN2HDAC1HDAC7
SCHEMBL18196803 0.78 ALDH1A1 (0.49) CYP3A4TDP1L3MBTL1MEN1KMT2A
SCHEMBL28515555 0.78 SLC15A1 (0.49) CYP3A4TDP1L3MBTL1CDC25BMEN1
SCHEMBL17164459 0.78 ALDH1A1 (0.46) RAB9ACYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL25981312 0.77 ALDH1A1 (0.51) CYP3A4TDP1L3MBTL1MEN1KMT2A
SCHEMBL17469040 0.77 ALDH1A1 (0.51) CYP3A4TDP1L3MBTL1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0010893-B1 ANTISECRETORY BRANCHED-CHAIN HETEROCYCLIC GUANIDINE DERIVATIVES, PROCESSES FOR THEIR MANUFACTURE, INTERMEDIATES, AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAID DERIVATIVES IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1984-02-08 EP disclosed
EP-0010893-A1 Antisecretory branched-chain heterocyclic guanidine derivatives, processes for their manufacture, intermediates, and pharmaceutical compositions containing said derivatives IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1980-05-14 EP disclosed