SCHEMBL11096016

SCHEMBL11096016

N#CC(CCC(=O)O)(CCC(=O)O)c1c(Cl)cccc1Cl

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 1/20 0.41
KMT2A Q03164 2/20 0.38
FFAR1 O14842 4/20 0.35
GPR17 Q13304 1/20 0.35
KDM4E B2RXH2 1/20 0.35
TSHR P16473 1/20 0.33
MEN1 O00255 1/20 0.33
FEN1 P39748 1/20 0.33
ALDH1A1 P00352 2/20 0.33
ESR1 P03372 1/20 0.33
CYP3A4 P08684 1/20 0.33
ESR2 Q92731 1/20 0.33
NOTUM Q6P988 1/20 0.32
AKR1B10 O60218 1/20 0.32
UGT1A9 O60656 1/20 0.32
TRPA1 O75762 1/20 0.32
ABCB11 O95342 1/20 0.32
MT-CO2 P00403 1/20 0.32
TTR P02766 1/20 0.32
ALB P02768 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7353916 0.91 AKR1B1 (0.37) AKR1B1KMT2AFFAR1GPR17KDM4E
SCHEMBL11818697 0.84 AKR1B1 (0.32) AKR1B1KMT2AKDM4EMEN1ALDH1A1
SCHEMBL11097563 0.83 FFAR1 (0.38) AKR1B1KMT2AFFAR1TSHRALDH1A1
SCHEMBL11818684 0.80 NLRP3 (0.43) KMT2AMEN1ALDH1A1
SCHEMBL11818689 0.79 EPHX2 (0.36) KMT2AKDM4EMEN1ALDH1A1CYP3A4
SCHEMBL8180989 0.77 KIF11 (0.40) KMT2AKDM4ETSHRMEN1FEN1
SCHEMBL11075302 0.76 CYP2C19 (0.40) FFAR1TSHRALDH1A1ESR1CYP3A4
SCHEMBL11066784 0.75 MIF (0.47) KMT2AFFAR1KDM4ETSHRMEN1
SCHEMBL6139367 0.75 TSHR (0.38) FFAR1TSHRALDH1A1ESR1CYP3A4
SCHEMBL11823090 0.75 MEN1 (0.31) AKR1B1KMT2AKDM4ETSHRMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4460604-A ANALGESICS, NARCOTIC ANTAGONIST THE UPJOHN COMPANY (US) 1984-07-17 US disclosed
US-4180584-A ANALGESIC; NARCOTIC ANTAGONIST THE UPJOHN COMPANY (US) 1979-12-25 US disclosed
US-4065573-A ANALGESICS THE UPJOHN COMPANY (US) 1977-12-27 US disclosed