SCHEMBL11097563

SCHEMBL11097563

N#CC(CCC(=O)O)(CCC(=O)O)c1ccccc1Cl

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FFAR1 O14842 3/20 0.38
HTR2A P28223 1/20 0.36
HTR2C P28335 1/20 0.36
ADRA1A P35348 1/20 0.36
OPRK1 P41145 1/20 0.36
KCNH2 Q12809 1/20 0.36
KIF11 P52732 1/20 0.36
AKR1B1 P15121 1/20 0.36
ALDH1A1 P00352 2/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2D6 P10635 1/20 0.35
TSHR P16473 1/20 0.35
CYP2C19 P33261 1/20 0.35
KCNN4 O15554 1/20 0.35
PTGFR P43088 3/20 0.34
KEAP1 Q14145 1/20 0.34
PTGS2 P35354 1/20 0.34
PTGDR2 Q9Y5Y4 2/20 0.33
HTT P42858 1/20 0.33
KMT2A Q03164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11093241 0.87 PTGFR (0.34) FFAR1HTR2AHTR2CADRA1AOPRK1
SCHEMBL11096016 0.83 AKR1B1 (0.41) FFAR1ADRA1AAKR1B1ALDH1A1TSHR
SCHEMBL11093234 0.82 ALDH1A1 (0.39) ALDH1A1TSHRHTTKMT2A
SCHEMBL21632134 0.82 HTR2A (0.38) FFAR1HTR2AHTR2CADRA1AOPRK1
SCHEMBL11092174 0.82 TDP1 (0.40) FFAR1ALDH1A1TSHR
SCHEMBL11093239 0.82 ALDH1A1 (0.34) ALDH1A1PTGFRHTTKMT2A
SCHEMBL8359862 0.81 KCNN4 (0.41) FFAR1ALDH1A1CYP1A2CYP2D6TSHR
SCHEMBL11103356 0.81 L3MBTL1 (0.39) FFAR1ALDH1A1CYP1A2CYP2D6TSHR
SCHEMBL11089297 0.80 FFAR1 (0.39) FFAR1AKR1B1ALDH1A1CYP1A2CYP2D6
SCHEMBL7128706 0.79 L3MBTL1 (0.43) FFAR1HTR2AHTR2CADRA1AOPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4460604-A ANALGESICS, NARCOTIC ANTAGONIST THE UPJOHN COMPANY (US) 1984-07-17 US disclosed
US-4180584-A ANALGESIC; NARCOTIC ANTAGONIST THE UPJOHN COMPANY (US) 1979-12-25 US disclosed
US-4065573-A ANALGESICS THE UPJOHN COMPANY (US) 1977-12-27 US disclosed