SCHEMBL11096038

SCHEMBL11096038

CC(CCc1ccccc1)NCc1ccccc1

nearest known ligand 0.81

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
BCHE P06276 2/20 0.71
SIGMAR1 Q99720 1/20 0.66
ATM Q13315 2/20 0.60
OPRK1 P41145 1/20 0.60
GAA P10253 1/20 0.60
KMT2A Q03164 4/20 0.57
ALDH1A1 P00352 3/20 0.57
SMN1; SMN2 Q16637 2/20 0.57
KCNH2 Q12809 1/20 0.54
TMEM97 Q5BJF2 1/20 0.54
L3MBTL1 Q9Y468 1/20 0.54
MEN1 O00255 3/20 0.53
CYP1A2 P05177 1/20 0.53
CYP2C9 P11712 1/20 0.53
CYP2C19 P33261 1/20 0.53
HTT P42858 1/20 0.53
HPGD P15428 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10451642 1.00 BCHE (0.71) BCHESIGMAR1ATMOPRK1GAA
SCHEMBL11816814 0.91 BCHE (0.67) BCHESIGMAR1ATMOPRK1GAA
SCHEMBL11815017 0.90 OPRK1 (0.77) BCHESIGMAR1ATMOPRK1GAA
SCHEMBL11535612 0.90 BCHE (0.65) BCHESIGMAR1ATMOPRK1GAA
SCHEMBL11824647 0.87 BCHE (0.74) BCHESIGMAR1ATMGAAKMT2A
SCHEMBL28983267 0.86 BCHE (0.60) BCHESIGMAR1ATMOPRK1GAA
SCHEMBL172531 0.84 SIGMAR1 (0.66) BCHESIGMAR1ATMOPRK1GAA
SCHEMBL13911191 0.84 SIGMAR1 (0.66) BCHESIGMAR1OPRK1KMT2AALDH1A1
SCHEMBL19498803 0.84 OPRK1 (0.81) BCHESIGMAR1OPRK1KMT2AALDH1A1
SCHEMBL14198232 0.84 SIGMAR1 (0.66) BCHESIGMAR1OPRK1KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117756659-A Preparation method of labetalol hydrochloride 重庆圣华曦药业股份有限公司 2024-03-26 CN disclosed
US-4450115-A ADRENERGIC BLOCKING AGENTS; HYPOTENSIVE AND CARDIOTONIC AGENTS KYOWA HAKKO KOGYO CO., LTD. (JP) 1984-05-22 US disclosed
US-4381398-A Amino-alcohol derivatives KYOWA HAKKO KOGYO CO., LTD. (JP) 1983-04-26 US disclosed
US-4217305-A HYPOTENSIVE AGENTS, ADRENERGIC BLOCKING AGENTS YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 1980-08-12 US disclosed
US-4140713-A Phenylethanolamine therapeutic agents ALLEN & HANBURYS LIMITED (GB) 1979-02-20 US disclosed
US-3943254-A ALPHA-AMINOMETHYL-4-HYDROXY-3-SULFAMYL BENZYL ALCOHOLS OR 4-HYDROXY-3-SULFAMYL-PHENETHYLAMINE SMITHKLINE CORPORATION (US) 1976-03-09 US disclosed