SCHEMBL11099237

SCHEMBL11099237

O=C1Nc2ccccc2CN1C1CCN(CC(O)c2ccc3c(c2)OCO3)CC1

nearest known ligand 0.55

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CTSS P25774 8/20 0.43
LMNA P02545 2/20 0.43
CHRM4 P08173 2/20 0.43
MAPK1 P28482 1/20 0.43
ALDH1A1 P00352 1/20 0.42
TSHR P16473 1/20 0.42
CHRM1 P11229 1/20 0.42
CALCRL Q16602 5/20 0.41
RAMP1 O60894 1/20 0.41
OPRM1 P35372 1/20 0.40
OPRD1 P41143 1/20 0.40
OPRK1 P41145 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11104912 0.85 LMNA (0.39) CTSSLMNAMAPK1ALDH1A1TSHR
SCHEMBL11108061 0.84 LMNA (0.43) LMNAMAPK1ALDH1A1TSHROPRM1
SCHEMBL11101376 0.84 CHRM4 (0.52) CTSSCHRM4CHRM1CALCRLRAMP1
SCHEMBL11105185 0.84 CTSS (0.57) CTSSCHRM4CHRM1CALCRLRAMP1
SCHEMBL11108153 0.82 CTSS (0.51) CTSSCHRM4TSHRCHRM1CALCRL
SCHEMBL11103893 0.82 CTSS (0.51) CTSSCHRM4CHRM1CALCRLRAMP1
SCHEMBL11102366 0.81 SCN1A (0.50) CTSSCHRM4CHRM1CALCRL
SCHEMBL11104105 0.80 MAOB (0.53) CTSSLMNACHRM4MAPK1ALDH1A1
SCHEMBL11099726 0.80 SCN1A (0.55) CTSSCHRM4CHRM1CALCRL
SCHEMBL11267525 0.79 LMNA (0.46) CTSSLMNAMAPK1ALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0029707-B1 NOVEL PIPERIDINE DERIVATIVES, METHOD FOR THE PREPARATION THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM KYOWA HAKKO KOGYO CO., LTD (JP) 1984-02-01 EP disclosed
US-4344948-A HYPOTENSIVE AGENTS KYOWA HAKKO KOGYO CO., LTD. (JP) 1982-08-17 US disclosed
EP-0029707-A1 Novel piperidine derivatives, method for the preparation thereof and pharmaceutical compositions containing them KYOWA HAKKO KOGYO CO., LTD (JP) 1981-06-03 EP disclosed