SCHEMBL11099532

SCHEMBL11099532

O=C(C=CC(c1ccc(Cl)cc1)N1C(=O)c2ccccc2C1=O)c1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOB P27338 2/20 0.47
CYP1B1 Q16678 1/20 0.43
LMNA P02545 2/20 0.43
MAPT P10636 4/20 0.41
ALDH1A1 P00352 2/20 0.41
HTT P42858 2/20 0.41
NPSR1 Q6W5P4 1/20 0.41
RECQL P46063 1/20 0.40
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
MAPK1 P28482 2/20 0.38
MMP2 P08253 1/20 0.38
MMP9 P14780 1/20 0.38
TNF P01375 1/20 0.38
CES2 O00748 1/20 0.37
CES1 P23141 1/20 0.37
KDM4E B2RXH2 1/20 0.37
APAF1 O14727 1/20 0.37
MITF O75030 1/20 0.37
POLB P06746 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30342198 0.72 TP53 (0.52) LMNAALDH1A1RECQLMEN1KMT2A
SCHEMBL29005218 0.72 TP53 (0.52) LMNAALDH1A1RECQLMEN1KMT2A
SCHEMBL4029880 0.71 ALOX15 (0.50) LMNAMAPTHTTNPSR1RECQL
SCHEMBL29130643 0.70 MAOB (0.72) MAOBCYP1B1LMNAMAPTALDH1A1
SCHEMBL17916031 0.70 DRD3 (0.52) MAPTALDH1A1NPSR1RECQLMEN1
SCHEMBL12846303 0.67 KMT2A (0.55) LMNAMAPTMEN1KMT2ATNF
SCHEMBL3462808 0.67 ALDH1A1 (0.47) MAOBCYP1B1LMNAMAPTALDH1A1
SCHEMBL3462807 0.67 ALDH1A1 (0.47) MAOBCYP1B1LMNAMAPTALDH1A1
SCHEMBL12845880 0.67 KMT2A (0.55) LMNAMAPTMEN1KMT2ATNF
SCHEMBL15664132 0.66 KMT2A (0.48) ALDH1A1RECQLMEN1KMT2ATNF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0045520-B1 PYRIMIDO-(4,5-D)(2)-BENZAZEPINES, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft (CH) 1984-06-20 EP disclosed