SCHEMBL11099657

SCHEMBL11099657

Clc1cc(C(Cl)(Cl)Cl)nc2c(-c3cccc4c(Cl)cc(C(Cl)(Cl)Cl)nc34)cccc12

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CRHR1 P34998 5/20 0.49
L3MBTL1 Q9Y468 2/20 0.43
CCR1 P32246 1/20 0.43
CCR8 P51685 1/20 0.43
CYP3A4 P08684 2/20 0.41
TSHR P16473 1/20 0.41
ENPP1 P22413 3/20 0.37
CYP1A2 P05177 2/20 0.37
CYP2A6 P11509 2/20 0.37
MAPT P10636 3/20 0.37
NR4A2 P43354 1/20 0.37
PARP1 P09874 1/20 0.36
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
APOBEC3G Q9HC16 1/20 0.35
ALDH1A1 P00352 2/20 0.35
KDM4E B2RXH2 1/20 0.35
MEN1 O00255 1/20 0.35
ALOX15B O15296 1/20 0.35
NR1I2 O75469 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9493152 0.89 NR4A2 (0.46) CRHR1L3MBTL1CCR1CCR8CYP3A4
SCHEMBL9492503 0.84 CYP3A4 (0.40) CRHR1L3MBTL1CCR1CCR8CYP3A4
SCHEMBL9492598 0.83 ELANE (0.44) CRHR1L3MBTL1CYP3A4TSHRMAPT
SCHEMBL21144535 0.83 MAPT (0.39) L3MBTL1CCR1CCR8CYP3A4TSHR
SCHEMBL9493489 0.81 ALDH1A1 (0.43) L3MBTL1CYP3A4TSHRCYP1A2PARP1
SCHEMBL10506369 0.81 CYP3A4 (0.38) CRHR1L3MBTL1CCR1CCR8CYP3A4
SCHEMBL9493850 0.80 LMNA (0.38) CRHR1L3MBTL1CCR1CCR8CYP3A4
SCHEMBL10824099 0.80 CYP3A4 (0.37) CRHR1L3MBTL1CCR1CCR8CYP3A4
SCHEMBL9494545 0.79 NQO2 (0.48) MAPTPARP1ALDH1A1KDM4EMEN1
SCHEMBL2710931 0.76 NT5E (0.48) L3MBTL1CCR1CCR8ENPP1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0113432-A1 Chloromethyl quinoline derivatives, process for their preparation and their use ALKALOIDA VEGYéSZETI GYáR (HU) 1984-07-18 EP claimed