SCHEMBL11100697

SCHEMBL11100697

CC(=O)CCCn1nc(-c2ccc(N(C)C)cc2)c(-c2ccc(N(C)C)cc2)nc1=O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
ACHE P22303 10/20 0.41
BACE1 P56817 10/20 0.41
MCHR1 Q99705 1/20 0.40
PTGIR P43119 1/20 0.37
KDM4E B2RXH2 1/20 0.36
TSHR P16473 1/20 0.36
HSD17B10 Q99714 1/20 0.36
PTGDR2 Q9Y5Y4 1/20 0.35
NPC1 O15118 1/20 0.35
ALDH1A1 P00352 1/20 0.35
CRHBP P24387 1/20 0.35
RAB9A P51151 1/20 0.35
CRHR2 Q13324 1/20 0.35
HDAC3 O15379 2/20 0.35
HDAC4 P56524 2/20 0.35
HDAC1 Q13547 2/20 0.35
HDAC7 Q8WUI4 2/20 0.35
HDAC2 Q92769 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11100991 0.85 MEN1 (0.50) MEN1KMT2AACHEBACE1PTGIR
SCHEMBL11096806 0.83 MEN1 (0.44) MEN1KMT2AACHEBACE1PTGIR
SCHEMBL11098924 0.75 KMT2A (0.54) MEN1KMT2AACHEBACE1
Metrazifone SCHEMBL2108915 0.74 NPC1 (0.43) MEN1KMT2AKDM4ETSHRHSD17B10
SCHEMBL11092723 0.71 ALPL (0.43) MEN1KMT2AACHEBACE1
SCHEMBL11096866 0.71 KDM5B (0.39) MEN1KMT2AKDM4EHSD17B10PTGDR2
SCHEMBL9770984 0.69 PTGIR (0.64) MEN1KMT2AACHEBACE1PTGIR
SCHEMBL9770992 0.69 PTGIR (0.64) MEN1KMT2AACHEBACE1PTGIR
SCHEMBL9770961 0.68 KMT2A (0.57) MEN1KMT2AACHEBACE1PTGIR
SCHEMBL5702986 0.66 ALDH1A1 (0.55) MEN1KMT2ATSHRHSD17B10NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0036357-B1 ANTALGIC AND ANTIAGREGANT CETONIC DERIVATIVES OF 5,6-DIARYL-1,2,4-TRIAZINES, USABLE IN THE TREATMENT OF MIGRAINE PIERRE FABRE S.A. (FR) 1984-05-30 EP claimed