SCHEMBL11101736

SCHEMBL11101736

COc1ccc2c(c1)CC[C@H]1[C@@H]2[C@H](C)C[C@]2(C)C(=O)CC[C@@H]12

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B1 P14061 3/20 0.67
LMNA P02545 2/20 0.67
MAPT P10636 2/20 0.67
RECQL P46063 1/20 0.67
SMN1; SMN2 Q16637 1/20 0.67
AKR1C3 P42330 3/20 0.60
KDM4E B2RXH2 2/20 0.54
HSD17B10 Q99714 2/20 0.54
TSHR P16473 1/20 0.54
MAPK1 P28482 1/20 0.54
STS P08842 6/20 0.53
ESR1 P03372 3/20 0.52
ESR2 Q92731 2/20 0.52
ABCC4 O15439 1/20 0.52
CYP2C9 P11712 1/20 0.52
ABCC1 P33527 1/20 0.52
SLCO1B1 Q9Y6L6 1/20 0.52
CA1 P00915 1/20 0.52
CA2 P00918 1/20 0.52
CA4 P22748 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9746964 0.88 HSD17B1 (0.66) HSD17B1LMNAMAPTRECQLSMN1; SMN2
SCHEMBL9634078 0.88 LMNA (0.66) HSD17B1LMNAMAPTRECQLSMN1; SMN2
SCHEMBL10531128 0.88 LMNA (0.66) HSD17B1LMNAMAPTRECQLSMN1; SMN2
SCHEMBL6468077 0.86 LMNA (0.64) HSD17B1LMNAMAPTRECQLSMN1; SMN2
SCHEMBL6465770 0.86 LMNA (0.64) HSD17B1LMNAMAPTRECQLSMN1; SMN2
SCHEMBL11101794 0.86 LMNA (0.64) HSD17B1LMNAMAPTRECQLSMN1; SMN2
SCHEMBL13930475 0.86 AKR1C3 (0.61) HSD17B1LMNAMAPTRECQLSMN1; SMN2
SCHEMBL17525935 0.85 LMNA (0.62) HSD17B1LMNAMAPTRECQLSMN1; SMN2
SCHEMBL14569770 0.84 HSD17B10 (0.70) HSD17B1LMNAMAPTRECQLSMN1; SMN2
SCHEMBL13930476 0.84 HSD17B10 (0.70) HSD17B1LMNAMAPTRECQLSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0044105-B1 NEW 8-ALPHA-OESTRA-1,3,5(10)-TRIENE DERIVATIVES, PROCESSES FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS AKZO N.V. (NL) 1984-10-03 EP claimed
EP-0044105-B1 NEW 8-ALPHA-OESTRA-1,3,5(10)-TRIENE DERIVATIVES, PROCESSES FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS AKZO N.V. (NL) 1984-10-03 EP disclosed
US-4407753-A 8α-Oestra-1,3,5(10)-triene derivatives, processes for their preparation and pharmaceutical compositions AKZO N.V. (NL) 1983-10-04 US disclosed
EP-0044105-A2 New 8-alpha-oestra-1,3,5(10)-triene derivatives, processes for their preparation and pharmaceutical compositions AKZO N.V. (NL) 1982-01-20 EP disclosed