SCHEMBL11109697

SCHEMBL11109697

CC(=O)n1cc2c3c(ccc(Cl)c31)C(O)C(NC(=O)CCl)C2

nearest known ligand 0.34

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 2/20 0.34
MTNR1B P49286 2/20 0.34
CNR1 P21554 2/20 0.33
SIGMAR1 Q99720 2/20 0.32
PYGL P06737 2/20 0.31
ALDH1A1 P00352 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11109699 1.00 MTNR1A (0.34) MTNR1AMTNR1BCNR1SIGMAR1PYGL
SCHEMBL11109702 1.00 MTNR1A (0.34) MTNR1AMTNR1BCNR1SIGMAR1PYGL
SCHEMBL11117091 0.77 ALDH1A1 (0.33) MTNR1AMTNR1BALDH1A1
SCHEMBL10669378 0.65 MTNR1A (0.40) MTNR1AMTNR1BPYGLALDH1A1
SCHEMBL697600 0.62 ALDH1A1 (0.60) MTNR1AMTNR1BALDH1A1
SCHEMBL696008 0.62 ALDH1A1 (0.60) MTNR1AMTNR1BALDH1A1
SCHEMBL696007 0.62 ALDH1A1 (0.60) MTNR1AMTNR1BALDH1A1
SCHEMBL697601 0.62 ALDH1A1 (0.60) MTNR1AMTNR1BALDH1A1
SCHEMBL7279700 0.62 ALDH1A1 (0.60) MTNR1AMTNR1BALDH1A1
SCHEMBL11272560 0.59 ALDH1A1 (0.42) MTNR1AMTNR1BALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0033767-B1 INDOLOBENZOXAZINES, PROCESSES FOR PREPARING AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME MERCK & CO. INC. (US) 1984-06-27 EP disclosed
US-4238486-A TREATING HYPERTENSION AND PARKINSON*S DISEASE MERCK & CO., INC. (US) 1980-12-09 US disclosed