SCHEMBL11117091

SCHEMBL11117091

CC(=O)n1cc2c3c(ccc(Cl)c31)C(=O)C(NC(=O)CCl)C2

nearest known ligand 0.33

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.33
MTNR1A P48039 1/20 0.32
MTNR1B P49286 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11110418 0.78 NOTUM (0.31) ALDH1A1
SCHEMBL11109699 0.77 MTNR1A (0.34) ALDH1A1MTNR1AMTNR1B
SCHEMBL11109702 0.77 MTNR1A (0.34) ALDH1A1MTNR1AMTNR1B
SCHEMBL11109697 0.77 MTNR1A (0.34) ALDH1A1MTNR1AMTNR1B
SCHEMBL11112840 0.71 NOTUM (0.35) ALDH1A1
SCHEMBL10681398 0.63 ALDH1A1 (0.41) ALDH1A1MTNR1AMTNR1B
SCHEMBL695898 0.59 SMN1; SMN2 (0.59) ALDH1A1MTNR1AMTNR1B
SCHEMBL696936 0.56 MAOB (0.46) ALDH1A1
SCHEMBL8312673 0.54 CYP11B1 (0.36)
SCHEMBL24614086 0.53 CYP19A1 (0.51) ALDH1A1MTNR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0033767-B1 INDOLOBENZOXAZINES, PROCESSES FOR PREPARING AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME MERCK & CO. INC. (US) 1984-06-27 EP disclosed
EP-0033767-A1 Indolobenzoxazines, processes for preparing and pharmaceutical compositions containing the same MERCK & CO. INC. (US) 1981-08-19 EP disclosed
US-4238486-A TREATING HYPERTENSION AND PARKINSON*S DISEASE MERCK & CO., INC. (US) 1980-12-09 US disclosed