SCHEMBL11113767

SCHEMBL11113767

COc1cccc(OCC(O)CN2CCC(c3c[nH]c4ccccc34)CC2)c1

nearest known ligand 0.62

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.59
TP53 P04637 2/20 0.56
MAPT P10636 2/20 0.56
KMT2A Q03164 1/20 0.56
SCN1A P35498 1/20 0.55
SCN5A Q14524 1/20 0.55
SCN9A Q15858 1/20 0.55
L3MBTL1 Q9Y468 1/20 0.55
HTR1A P08908 5/20 0.53
KDM4E B2RXH2 1/20 0.52
MAPK1 P28482 1/20 0.51
ADRB2 P07550 1/20 0.51
ADRB1 P08588 1/20 0.51
ADRB3 P13945 1/20 0.51
SMN1; SMN2 Q16637 1/20 0.50
SLC6A4 P31645 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL11007073 0.90 GAA (0.59) GAAMAPTKMT2AL3MBTL1HTR1A
SCHEMBL11117325 0.90 KMT2A (0.57) KMT2AHTR1ASMN1; SMN2SLC6A4
SCHEMBL11118598 0.88 KMT2A (0.53) GAAKMT2AL3MBTL1HTR1AMAPK1
SCHEMBL11010053 0.82 DRD4 (0.64) MAPTKMT2AHTR1AKDM4EMAPK1
Hydrochloric Acid SCHEMBL11015770 0.81 LMNA (0.64) MAPTKMT2AHTR1AKDM4EADRB2
SCHEMBL7079931 0.79 KMT2A (0.56) GAAMAPTKMT2AL3MBTL1HTR1A
SCHEMBL10784748 0.79 HTR1A (0.51) MAPTKMT2AHTR1AADRB2ADRB1
Hydrochloric Acid SCHEMBL11013120 0.79 KMT2A (0.60) KMT2AHTR1AADRB2ADRB1ADRB3
Hydrochloric Acid SCHEMBL11014416 0.79 KMT2A (0.60) MAPTKMT2AHTR1AKDM4EMAPK1
Hydrochloric Acid SCHEMBL11010332 0.79 HTR1A (0.50) GAAMAPTKMT2AHTR1AADRB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0112191-A1 4-(1H-indolyl-3-)-alpha-methyl piperidine-1-ethanol derivatives, their salts, process for their preparation, compositions containing them and their use as medicines ROUSSEL-UCLAF (FR) 1984-06-27 EP disclosed