SCHEMBL11116056

SCHEMBL11116056

Cc1ccc(C(O)(CCN(C)CCN(C)Cc2ccccc2)c2ccccc2)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.53
CHRM2 P08172 1/20 0.52
CHRM4 P08173 1/20 0.52
CHRM5 P08912 1/20 0.52
CHRM1 P11229 1/20 0.52
CHRM3 P20309 1/20 0.52
MEN1 O00255 5/20 0.49
KMT2A Q03164 5/20 0.49
BCL2 P10415 1/20 0.45
CARM1 Q86X55 1/20 0.44
PRMT6 Q96LA8 1/20 0.44
PRMT8 Q9NR22 1/20 0.44
HTR2A P28223 1/20 0.42
HTR2C P28335 1/20 0.42
ADRA1A P35348 1/20 0.42
OPRK1 P41145 1/20 0.42
KCNH2 Q12809 1/20 0.42
SIGMAR1 Q99720 4/20 0.41
NPSR1 Q6W5P4 2/20 0.41
ALDH1A1 P00352 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11112967 0.93 SMN1; SMN2 (0.60) SMN1; SMN2CHRM2CHRM4CHRM5CHRM1
SCHEMBL11114118 0.90 TSHR (0.52) SMN1; SMN2CHRM2CHRM4CHRM5CHRM1
SCHEMBL11114288 0.88 BCL2 (0.60) SMN1; SMN2CHRM2CHRM4CHRM5CHRM1
SCHEMBL11115170 0.85 TSHR (0.56) SMN1; SMN2CHRM2CHRM4CHRM5CHRM1
SCHEMBL11125959 0.84 SMN1; SMN2 (0.57) SMN1; SMN2CHRM2CHRM4CHRM5CHRM1
SCHEMBL9750628 0.84 TSHR (0.57) SMN1; SMN2CHRM2CHRM4CHRM5CHRM1
SCHEMBL11110419 0.81 SIGMAR1 (0.55) SMN1; SMN2CHRM2CHRM4CHRM5CHRM1
SCHEMBL11116143 0.80 SMN1; SMN2 (0.51) SMN1; SMN2CHRM2CHRM4CHRM5CHRM1
SCHEMBL11111482 0.79 LMNA (0.52) SMN1; SMN2CHRM2CHRM4CHRM5CHRM1
SCHEMBL11109990 0.79 TSHR (0.51) SMN1; SMN2CHRM2CHRM4CHRM5CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0041757-B1 ETHYLENDIAMINE DERIVATIVES, PREPARATION THEREOF, PHARMACEUTICAL COMPOSITIONS CONTAINING SAME AND INTERMEDIATES FOR THEIR PREPARATION Simes S.p.A. (IT) 1984-11-07 EP disclosed