SCHEMBL11116090

SCHEMBL11116090

CC(Br)C(=O)c1ccc(CCCO)c(Cl)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2C9 P11712 1/20 0.39
SLC6A4 P31645 4/20 0.36
SLC6A3 Q01959 4/20 0.36
SLC6A2 P23975 3/20 0.36
CHRNA1 P02708 1/20 0.36
CHRNG P07510 1/20 0.36
CHRNB1 P11230 1/20 0.36
CHRNB2 P17787 1/20 0.36
CHRNB4 P30926 1/20 0.36
CHRNA3 P32297 1/20 0.36
CHRNA4 P43681 1/20 0.36
CHRND Q07001 1/20 0.36
HPGD P15428 2/20 0.35
KDM4E B2RXH2 1/20 0.35
DBH P09172 1/20 0.35
GAA P10253 1/20 0.35
RECQL P46063 1/20 0.35
CYP4A11 Q02928 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11108767 0.80 SLC6A3 (0.62) ALDH1A1SLC6A4SLC6A3SLC6A2CHRNA1
Hydrochloric Acid SCHEMBL11115575 0.79 SLC6A3 (0.61) ALDH1A1SLC6A4SLC6A3SLC6A2CHRNA1
SCHEMBL11109327 0.78 MAPT (0.41) ALDH1A1HPGDCYP4A11TAS1R3TAS1R1
SCHEMBL633270 0.76 TSHR (0.53) ALDH1A1CYP1A2CYP2C9SLC6A4SLC6A3
SCHEMBL11113373 0.76 ALDH1A1 (0.38) ALDH1A1CYP1A2CYP2C9SLC6A4SLC6A3
SCHEMBL12438197 0.73 KDM4E (0.50) SLC6A4SLC6A3SLC6A2CHRNA1CHRNG
SCHEMBL634550 0.73 SLC6A2 (0.60) ALDH1A1CYP1A2CYP2C9SLC6A4SLC6A3
SCHEMBL786551 0.72 SMN1; SMN2 (0.51) ALDH1A1CYP1A2CYP2C9SLC6A4SLC6A3
SCHEMBL4104239 0.72 SLC6A2 (0.46) ALDH1A1CYP1A2CYP2C9SLC6A4SLC6A3
SCHEMBL5937704 0.72 KDM4E (0.52) SLC6A4SLC6A3SLC6A2CHRNA1CHRNG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0038071-B1 NEW UNLABELLED AND RADIOACTIVE LABELLED DERIVATIVES OF BUTYLAMINO PROPIOPHENONE, THEIR PREPARATION, IMMUNOGENS OBTAINED FROM THE UNLABELLED DERIVATIVES AND A PROCESS FOR IMMUNOGEN PREPARATION, ANTISERA RAISED USING THE IMMUNOGENS AND A METHOD FOR RAISING ANTISERA, A RADIOIMMUNOASSAY METHOD AND A TEST KIT FOR USE IN THE ASSAY METHOD THE WELLCOME FOUNDATION LIMITED (GB) 1984-11-14 EP disclosed
US-4356165-A Bupropion radioimmunoassay, and kit BURROUGHS WELLCOME CO. (US) 1982-10-26 US disclosed
US-4355179-A Radioactive nuclide labeled propiophenone compounds BURROUGHS WELLCOME CO. (US) 1982-10-19 US disclosed
US-4347177-A Compounds and methods of making them BURROUGHS WELLCOME CO. (US) 1982-08-31 US disclosed
US-4347382-A 3H Labeled compounds BURROUGHS WELLCOME CO. (US) 1982-08-31 US disclosed
US-4347178-A Compounds and methods of making BURROUGHS WELLCOME CO. (US) 1982-08-31 US disclosed
US-4347176-A Compounds and methods of making same BURROUGHS WELLCOME CO. (US) 1982-08-31 US disclosed
EP-0038071-A2 New unlabelled and radioactive labelled derivatives of butylamino propiophenone, their preparation, immunogens obtained from the unlabelled derivatives and a process for immunogen preparation, antisera raised using the immunogens and a method for raising antisera, a radioimmunoassay method and a test kit for use in the assay method THE WELLCOME FOUNDATION LIMITED (GB) 1981-10-21 EP disclosed