SCHEMBL11117589

SCHEMBL11117589

O=c1ncc2ccc3ncncc3c2[nH]1

nearest known ligand 0.34

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
EGFR P00533 9/20 0.34
PDE5A O76074 1/20 0.32
TDO2 P48775 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1982985 0.77 CYP3A4 (0.47)
SCHEMBL28575817 0.75 MAPT (0.40) EGFR
SCHEMBL30949930 0.75 MAPT (0.40) EGFR
SCHEMBL1808544 0.74 EGFR (0.38) EGFRTDO2
SCHEMBL30961886 0.74 EGFR (0.38) EGFRTDO2
SCHEMBL2811653 0.73 PKM (0.31)
SCHEMBL6903705 0.73 HPGD (0.54) TDO2
SCHEMBL1287815 0.73 MCL1 (0.46)
SCHEMBL9037556 0.72
SCHEMBL25278009 0.71 KDM4E (0.50)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4455312-A 2-(o-Carboxyphenylamino)-6H-pyrimido(2,1-b)-quinazolone-6 and derivatives thereof, and application as antiphlogistics KIEVSKY NAUCHNO-ISSLEDOVATELSKY INSTITUT FARMAKOLOGIII TOXIKOLOGII USSR. KIEV ULITSA EXHENA POTIE, 14 1984-06-19 US disclosed