SCHEMBL1114291

SCHEMBL1114291

Oc1c(Cl)cc(C2N=CN(Cc3cccc(OC(F)F)c3)O2)cc1Cl

nearest known ligand 0.35

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CETP P11597 4/20 0.35
P2RX7 Q99572 1/20 0.35
DAO P14920 1/20 0.35
HCRTR1 O43613 3/20 0.35
HCRTR2 O43614 3/20 0.35
KMT2A Q03164 1/20 0.35
KAT2B Q92831 1/20 0.35
MEP1B Q16820 1/20 0.34
SCN1A P35498 1/20 0.33
SCN8A Q9UQD0 1/20 0.33
ROCK2 O75116 2/20 0.33
ALKBH1 Q13686 1/20 0.33
KCNJ5 P48544 1/20 0.33
KCNJ3 P48549 1/20 0.33
THRA P10827 1/20 0.32
THRB P10828 1/20 0.32
P2RX3 P56373 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1114748 0.88 HSD17B13 (0.40) CETPP2RX7HCRTR1HCRTR2ROCK2
SCHEMBL1114304 0.78 HCRTR1 (0.36) CETPP2RX7DAOHCRTR1HCRTR2
SCHEMBL1114303 0.71 MEP1B (0.36) CETPP2RX7DAOHCRTR1HCRTR2
SCHEMBL1114292 0.69 MEP1B (0.36) CETPP2RX7DAOHCRTR1HCRTR2
SCHEMBL10913301 0.62 MEP1B (0.50) DAOHCRTR1HCRTR2KMT2AMEP1B
SCHEMBL1776057 0.62 MEP1B (0.54) DAOKMT2AMEP1BROCK2ALKBH1
SCHEMBL10697500 0.61 HSD17B10 (0.44) KMT2AKCNJ5KCNJ3THRB
SCHEMBL3247033 0.61 KMT2A (0.46) KMT2AROCK2
SCHEMBL4504413 0.60 FEN1 (0.39) CETPHCRTR1HCRTR2
SCHEMBL31010320 0.60 SMN1; SMN2 (0.58) KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2278879-A2 COMPOUNDS, COMPOSITIONS AND METHODS COMPRISING OXADIAZOLE DERIVATIVES Institute for OneWorld Health (US) 2011-02-02 EP claimed
WO-2009131957-A2 COMPOUNDS, COMPOSITIONS AND METHODS COMPRISING OXADIAZOLE DERIVATIVES INSTITUTE FOR ONEWORLD HEALTH (US) 2009-10-29 WO claimed
EP-2278879-A2 COMPOUNDS, COMPOSITIONS AND METHODS COMPRISING OXADIAZOLE DERIVATIVES Institute for OneWorld Health (US) 2011-02-02 EP disclosed
WO-2009131957-A2 COMPOUNDS, COMPOSITIONS AND METHODS COMPRISING OXADIAZOLE DERIVATIVES INSTITUTE FOR ONEWORLD HEALTH (US) 2009-10-29 WO disclosed