SCHEMBL1114587

SCHEMBL1114587

O=C(NCc1cccc(OC(F)(F)F)c1)c1nc(Cc2cc(Br)c(O)c(Br)c2)no1

nearest known ligand 0.49

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 5/20 0.48
ROCK1 Q13464 4/20 0.48
MAPK14 Q16539 1/20 0.48
KLKB1 P03952 1/20 0.44
GLS O94925 5/20 0.44
MMP13 P45452 1/20 0.43
ABCB1 P08183 1/20 0.41
NAMPT P43490 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1114331 0.86 ROCK2 (0.53) ROCK2ROCK1MAPK14GLSMMP13
SCHEMBL1114287 0.80 ROCK2 (0.52) ROCK2ROCK1MAPK14GLSMMP13
SCHEMBL1114286 0.76 SMN1; SMN2 (0.52)
SCHEMBL13447645 0.74 LMNA (0.54) ROCK2ROCK1MMP13
SCHEMBL3242530 0.72 SMN1; SMN2 (0.57) ROCK2ROCK1MAPK14
SCHEMBL1114987 0.72 ROCK2 (0.51) ROCK2ROCK1MAPK14GLSMMP13
SCHEMBL2318885 0.72 GLS (0.51) ROCK2ROCK1MAPK14GLSABCB1
SCHEMBL1114182 0.70 POLB (0.52)
SCHEMBL18352279 0.70 MAPK14 (0.58) ROCK2ROCK1MAPK14GLSMMP13
SCHEMBL29351167 0.70 MAPK14 (0.58) ROCK2ROCK1MAPK14GLSMMP13

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2278879-A2 COMPOUNDS, COMPOSITIONS AND METHODS COMPRISING OXADIAZOLE DERIVATIVES Institute for OneWorld Health (US) 2011-02-02 EP claimed
WO-2009131957-A2 COMPOUNDS, COMPOSITIONS AND METHODS COMPRISING OXADIAZOLE DERIVATIVES INSTITUTE FOR ONEWORLD HEALTH (US) 2009-10-29 WO claimed