SCHEMBL1114755

SCHEMBL1114755

CC1(Cc2ccc(OCCCCN3CCN(c4cccc(Cl)c4Cl)CC3)cc2)N=NN=N1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 16/20 0.59
HTR2A P28223 5/20 0.59
HTR1A P08908 3/20 0.59
DRD3 P35462 10/20 0.58
DRD4 P21917 4/20 0.58
KCNH2 Q12809 3/20 0.57
HTR3E A5X5Y0 1/20 0.54
MEN1 O00255 1/20 0.54
MLNR O43193 1/20 0.54
HTR3B O95264 1/20 0.54
ABCB11 O95342 1/20 0.54
ESR1 P03372 1/20 0.54
PGR P06401 1/20 0.54
ADRB2 P07550 1/20 0.54
CHRM2 P08172 1/20 0.54
ABCB1 P08183 1/20 0.54
ADRB1 P08588 1/20 0.54
ADRA2A P08913 1/20 0.54
ADORA3 P0DMS8 1/20 0.54
GAA P10253 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12403746 0.84 DRD2 (0.66) DRD2HTR2AHTR1ADRD3DRD4
SCHEMBL1114150 0.81 DRD2 (0.64) DRD2HTR2AHTR1ADRD3DRD4
SCHEMBL1114430 0.81 DRD2 (0.60) DRD2HTR2AHTR1ADRD3DRD4
SCHEMBL1114311 0.80 DRD2 (0.62) DRD2HTR2AHTR1ADRD3DRD4
SCHEMBL1114462 0.79 DRD2 (0.58) DRD2HTR2AHTR1ADRD3DRD4
SCHEMBL1114412 0.79 DRD2 (0.59) DRD2HTR2AHTR1ADRD3DRD4
SCHEMBL4244520 0.79 DRD2 (0.67) DRD2HTR2AHTR1ADRD3DRD4
SCHEMBL1114397 0.79 DRD2 (0.60) DRD2HTR2AHTR1ADRD3DRD4
SCHEMBL29771174 0.78 DRD2 (0.64) DRD2HTR2AHTR1ADRD3DRD4
SCHEMBL12403727 0.76 HRH3 (0.62) DRD2HTR2AHTR1ADRD3DRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2279179-A2 PHENYL PIPERAZINE COMPOUNDS, PHARMACEUTICAL COMPOSITION INCLUDING THE SAME, AND USE THEREOF SK Holdings Co., Ltd. (KR) 2011-02-02 EP claimed
WO-2009145591-A2 PHENYL PIPERAZINE COMPOUNDS, PHARMACEUTICAL COMPOSITION INCLUDING THE SAME, AND USE THEREOF SK HOLDINGS CO., LTD. (KR) 2009-12-03 WO claimed