SCHEMBL1114833

SCHEMBL1114833

Oc1c(Cl)cc(C2N=CON2Cc2ccccc2C(F)(F)F)cc1Cl

nearest known ligand 0.38

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HSD17B13 Q7Z5P4 8/20 0.38
KDM4E B2RXH2 2/20 0.36
ALDH1A1 P00352 2/20 0.36
ATM Q13315 1/20 0.36
P2RX7 Q99572 1/20 0.36
HSP90AA1 P07900 1/20 0.35
HSP90B1 P14625 1/20 0.35
STK10 O94804 1/20 0.34
SLK Q9H2G2 1/20 0.34
SIRT2 Q8IXJ6 1/20 0.34
SIRT1 Q96EB6 1/20 0.34
NR1H2 P55055 1/20 0.34
NR1H3 Q13133 1/20 0.34
NPBWR1 P48145 1/20 0.34
EPHX2 P34913 1/20 0.34
PPARG P37231 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1114610 0.87 ALDH1A1 (0.34) KDM4EALDH1A1ATMSIRT2SIRT1
SCHEMBL1114304 0.70 HCRTR1 (0.36) HSD17B13P2RX7
SCHEMBL4372432 0.68 HSD17B13 (0.43) HSD17B13KDM4EALDH1A1ATMP2RX7
SCHEMBL1114336 0.67 KDM4E (0.39) HSD17B13KDM4EALDH1A1ATMP2RX7
SCHEMBL4355638 0.67 UTS2R (0.51) HSD17B13KDM4EALDH1A1ATMP2RX7
SCHEMBL4359436 0.61 GAA (0.44) HSD17B13KDM4EALDH1A1P2RX7HSP90AA1
SCHEMBL1491106 0.61 KDM4E (0.46) KDM4EALDH1A1ATMP2RX7SIRT2
SCHEMBL3980590 0.59 KDM4E (0.53) KDM4EALDH1A1ATMP2RX7SIRT2
SCHEMBL28221686 0.58 ALDH1A1 (0.48) KDM4EALDH1A1ATMP2RX7NR1H2
SCHEMBL44837 0.57 IDO1 (0.57) KDM4EALDH1A1ATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2278879-A2 COMPOUNDS, COMPOSITIONS AND METHODS COMPRISING OXADIAZOLE DERIVATIVES Institute for OneWorld Health (US) 2011-02-02 EP disclosed
WO-2009131957-A2 COMPOUNDS, COMPOSITIONS AND METHODS COMPRISING OXADIAZOLE DERIVATIVES INSTITUTE FOR ONEWORLD HEALTH (US) 2009-10-29 WO disclosed