SCHEMBL11153646

SCHEMBL11153646

CCOC(=O)c1c(Cl)c2cnc(-c3ccccc3)nc2n(CC)c1=O

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.49
SMN1; SMN2 Q16637 5/20 0.49
MAPT P10636 3/20 0.49
LMNA P02545 3/20 0.49
MAPK1 P28482 1/20 0.49
ATM Q13315 1/20 0.49
L3MBTL1 Q9Y468 2/20 0.48
RAB9A P51151 4/20 0.48
KDM4E B2RXH2 4/20 0.48
NPC1 O15118 3/20 0.48
TP53 P04637 2/20 0.48
CYP1A2 P05177 4/20 0.47
POLB P06746 2/20 0.47
CYP2C9 P11712 2/20 0.46
CYP2C19 P33261 2/20 0.46
CSNK1D P48730 1/20 0.45
HSD17B10 Q99714 1/20 0.44
FOS P01100 2/20 0.43
JUN P05412 2/20 0.43
NFKB1 P19838 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11158393 0.89 LMNA (0.50) ALDH1A1SMN1; SMN2MAPTLMNAMAPK1
SCHEMBL11155574 0.89 L3MBTL1 (0.47) ALDH1A1SMN1; SMN2MAPTLMNAMAPK1
SCHEMBL11155855 0.89 KDM4E (0.60) ALDH1A1SMN1; SMN2MAPTLMNAMAPK1
SCHEMBL11161803 0.85 ALDH1A1 (0.47) ALDH1A1SMN1; SMN2MAPTLMNAMAPK1
SCHEMBL11158611 0.84 ALDH1A1 (0.47) ALDH1A1SMN1; SMN2MAPTLMNAMAPK1
SCHEMBL11157777 0.82 ADORA2A (0.45) ALDH1A1SMN1; SMN2MAPTLMNAMAPK1
SCHEMBL2087647 0.82 KDM4E (0.52) ALDH1A1SMN1; SMN2MAPTLMNAMAPK1
SCHEMBL11210201 0.81 ALDH1A1 (0.46) ALDH1A1SMN1; SMN2MAPTLMNAMAPK1
SCHEMBL11157510 0.81 KDM4E (0.53) ALDH1A1SMN1; SMN2MAPTLMNAMAPK1
SCHEMBL11158112 0.79 LMNA (0.61) ALDH1A1SMN1; SMN2MAPTLMNAMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4233446-A 5-Chloro-7,8-dihydro-7-oxo-pyrido[2,3-d]pyrimidine-6-carboxylic acid derivatives AMERICAN HOME PRODUCTS CORPORATION (US) 1980-11-11 US claimed
EP-0018139-B1 PYRIDO (2,3-D) PYRIMIDINE DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND PROCESSES FOR PREPARING THE PYRIDO (2,3-D) PYRIMIDINE DERIVATIVES AMERICAN HOME PRODUCTS CORPORATION (US) 1983-05-04 EP disclosed
US-4301281-A 7,8-Dihydro-2,5,8-trisubstituted-7-oxo-pyrido[2,3-d]-pyrimidine-6-carboxylic acid amides AMERICAN HOME PRODUCTS CORPORATION (US) 1981-11-17 US disclosed
US-4255568-A ANTIALLERGENS AND ANTISECRETORY AGENTS AMERICAN HOME PRODUCTS CORPORATION (US) 1981-03-10 US disclosed
US-4236004-A 2-Alkylsulphonyl-7,8-dihydro-5-hydroxy-7-oxo-pyrido[2,3-d]pyrimidine-6-carboxylic acid derivatives AMERICAN HOME PRODUCTS CORPORATION (US) 1980-11-25 US disclosed
US-4233446-A 5-Chloro-7,8-dihydro-7-oxo-pyrido[2,3-d]pyrimidine-6-carboxylic acid derivatives AMERICAN HOME PRODUCTS CORPORATION (US) 1980-11-11 US disclosed
EP-0018139-A2 Pyrido (2,3-d) pyrimidine derivatives, pharmaceutical compositions containing them and processes for preparing the pyrido (2,3-d) pyrimidine derivatives AMERICAN HOME PRODUCTS CORPORATION (US) 1980-10-29 EP disclosed
US-4215216-A 7,8-Dihydro-2,5,8-trisubstituted-7-oxo-pyrido[2,3-d]pyrimidine-6-carboxylic acid derivatives AMERICAN HOME PRODUCTS CORPORATION (US) 1980-07-29 US disclosed