SCHEMBL11173744

SCHEMBL11173744

CCOC(=O)Oc1nc2c3ccc(C(F)(F)F)cc3[nH]c(=O)n2n1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 1/20 0.44
PAK4 O96013 1/20 0.44
NTRK1 P04629 1/20 0.44
LCK P06239 1/20 0.44
FYN P06241 1/20 0.44
CSF1R P07333 1/20 0.44
RET P07949 1/20 0.44
MET P08581 1/20 0.44
PDGFRB P09619 1/20 0.44
PIM1 P11309 1/20 0.44
FGFR1 P11362 1/20 0.44
PRKACA P17612 1/20 0.44
GRK5 P34947 1/20 0.44
MAP2K2 P36507 1/20 0.44
FLT3 P36888 1/20 0.44
MAPK8 P45983 1/20 0.44
CDK8 P49336 1/20 0.44
GSK3A P49840 1/20 0.44
GSK3B P49841 1/20 0.44
CDK7 P50613 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8375789 0.86 CA12 (0.48) CA12CA9HAVCR2MAPTKIF11
SCHEMBL11085153 0.85 ADORA3 (0.50) ADORA3
SCHEMBL8376738 0.82 JAK2 (0.49) JAK2PAK4NTRK1LCKFYN
SCHEMBL11172982 0.82 HAVCR2 (0.60) JAK2PAK4NTRK1LCKFYN
SCHEMBL10924899 0.80 JAK2 (0.55) JAK2PAK4NTRK1LCKFYN
SCHEMBL11167343 0.80 GRIN1 (0.40) MAPTADORA3KIF11KDM4E
SCHEMBL462802 0.79 HAVCR2 (0.67) CA12CA9HAVCR2MAPTHSD17B10
SCHEMBL10924909 0.78 JAK2 (0.53) JAK2PAK4NTRK1LCKFYN
SCHEMBL11173600 0.77 JAK2 (0.45) JAK2PAK4NTRK1LCKFYN
SCHEMBL10927464 0.74 ADORA3 (0.41) JAK2PAK4NTRK1LCKFYN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0080176-A1 Triazoloquinazolines, process for their preparation and pharmaceutical compositions containing them BASF Aktiengesellschaft (DE) 1983-06-01 EP disclosed