SCHEMBL8375789

SCHEMBL8375789

O=C(O)Oc1nc2c3ccc(C(F)(F)F)cc3[nH]c(=O)n2n1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.48
CA9 Q16790 1/20 0.48
HAVCR2 Q8TDQ0 2/20 0.42
MEN1 O00255 2/20 0.41
CYP1A2 P05177 2/20 0.41
KMT2A Q03164 2/20 0.41
ALDH1A1 P00352 2/20 0.41
HPGD P15428 2/20 0.41
ALOX12 P18054 1/20 0.41
MAPT P10636 2/20 0.40
NFKB1 P19838 2/20 0.40
HSP90AA1 P07900 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2C9 P11712 1/20 0.40
TSHR P16473 1/20 0.40
CYP2C19 P33261 1/20 0.40
BLM P54132 1/20 0.40
PMP22 Q01453 1/20 0.40
KCNMA1 Q12791 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11173744 0.86 JAK2 (0.44) CA12CA9HAVCR2ALDH1A1HPGD
SCHEMBL11161587 0.83 HAVCR2 (0.50) HAVCR2ALDH1A1HPGDGABRPGABRD
SCHEMBL11167166 0.81 HAVCR2 (0.46) HAVCR2ALDH1A1HPGDGABRPGABRD
SCHEMBL10922730 0.80 GABRP (0.60) HAVCR2ALDH1A1HPGDGABRPGABRD
SCHEMBL8375791 0.79 PARP1 (0.41) CA12CA9HAVCR2ALDH1A1HPGD
SCHEMBL11085153 0.79 ADORA3 (0.50)
SCHEMBL462802 0.79 HAVCR2 (0.67) CA12CA9HAVCR2MAPTHSD17B10
SCHEMBL8376736 0.78 JAK2 (0.44) HAVCR2ALDH1A1HPGDKDM4EHSD17B10
SCHEMBL11170424 0.77 JAK2 (0.46) HAVCR2ALDH1A1HPGDGABRPGABRD
SCHEMBL11172659 0.77 JAK2 (0.43) HAVCR2ALDH1A1HPGDGABRPGABRD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0673249-B1 TRIAZOLOQUINAZOLINES FOR THE TREATMENT OF DISEASES OF THE CENTRAL NERVOUS SYSTEM BASF AG (DE) 1999-03-17 EP disclosed