SCHEMBL11178205

SCHEMBL11178205

Brc1ccc2[nH]cc(CNc3ccccc3)c2c1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR84 Q9NQS5 1/20 0.59
HTR2A P28223 2/20 0.54
TRPM8 Q7Z2W7 1/20 0.54
IDO1 P14902 1/20 0.53
CSNK2A1 P68400 1/20 0.52
HTR1A P08908 3/20 0.48
MTNR1A P48039 1/20 0.48
MTNR1B P49286 1/20 0.48
SLC6A4 P31645 3/20 0.48
SIGMAR1 Q99720 2/20 0.47
HRH3 Q9Y5N1 2/20 0.45
DRD2 P14416 2/20 0.45
DRD3 P35462 2/20 0.45
ADRA2A P08913 1/20 0.45
ADRA2B P18089 1/20 0.45
ADRA2C P18825 1/20 0.45
SLC6A2 P23975 1/20 0.45
ADRA1D P25100 1/20 0.45
HTR1D P28221 1/20 0.45
HTR1B P28222 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11173942 0.82 HTR2A (0.55) GPR84HTR2ATRPM8IDO1HTR1A
SCHEMBL5897571 0.81 HRH3 (0.60) GPR84HTR2AIDO1HTR1AHRH3
SCHEMBL17829924 0.81 GPR84 (0.54) GPR84HTR2ATRPM8IDO1CSNK2A1
SCHEMBL11180317 0.79 GPR84 (0.63) GPR84HTR2ATRPM8HTR1AHTR1D
SCHEMBL31415110 0.78 GPR84 (0.72) GPR84HTR2ATRPM8IDO1CSNK2A1
SCHEMBL28547448 0.77 GPR84 (0.75) GPR84HTR2ATRPM8IDO1CSNK2A1
SCHEMBL28972158 0.77 RAB9A (0.52) GPR84HTR2ATRPM8IDO1CSNK2A1
SCHEMBL3783656 0.76 HTR2A (0.65) GPR84HTR2ATRPM8CSNK2A1HTR1A
SCHEMBL12903067 0.76 GPR84 (0.63) GPR84HTR2ATRPM8IDO1CSNK2A1
SCHEMBL5430044 0.76 HTR2A (0.80) GPR84HTR2ATRPM8IDO1CSNK2A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4372887-A DIURETIC, ANTITHROMBOGENIC, SMOOTH MUSCLE RELAXANTS MEAD JOHNSON & COMPANY (US) 1983-02-08 US disclosed
US-4259238-A ANTIARRHYTHMIA AGENTS MEAD JOHNSON & COMPANY (US) 1981-03-31 US disclosed
US-4196212-A DIURETIC, ANTITHROMBOGENIC, SMOOTH MUSCLE RELAXANT, ANTIINFLAMMATORY MEAD JOHNSON & COMPANY (US) 1980-04-01 US disclosed
US-4072675-A DIURETICS, ANTICOAGULANTS, INOTROPIC AGENTS, ANTIINFLAMMATORY AGENTS, ANTIARRHYTHMIA AGENTS MEAD JOHNSON & COMPANY (US) 1978-02-07 US disclosed
US-4049714-A DIURETIC, ANTITHROMBOGENIC, ANTIARRYTHMIC, ANTIINFLAMMATORY, MUSCLE RELAXANTS MEAD JOHNSON & COMPANY (US) 1977-09-20 US disclosed