SCHEMBL11178299

SCHEMBL11178299

S=C=Nc1cccc2ccoc12

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.52
CYP3A4 P08684 2/20 0.52
TDP1 Q9NUW8 2/20 0.52
ALDH1A1 P00352 2/20 0.52
SLC6A4 P31645 2/20 0.52
ABCB11 O95342 1/20 0.52
NR3C1 P04150 1/20 0.52
ADRA2A P08913 1/20 0.52
ADORA3 P0DMS8 1/20 0.52
HPGD P15428 1/20 0.52
ALOX15 P16050 1/20 0.52
ADRA2C P18825 1/20 0.52
MAOA P21397 1/20 0.52
DRD1 P21728 1/20 0.52
HTR2B P41595 1/20 0.52
CCR2 P41597 1/20 0.52
HSD17B10 Q99714 1/20 0.52
MEN1 O00255 1/20 0.45
NPC1 O15118 1/20 0.45
CYP2D6 P10635 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27363685 0.70 MAOA (0.52) CYP1A2CYP3A4TDP1ALDH1A1SLC6A4
1-Naphthylisothiocyanate SCHEMBL29354904 0.68 ALDH1A1 (1.00) CYP1A2CYP3A4TDP1ALDH1A1SLC6A4
1-Naphthylisothiocyanate SCHEMBL419795 0.68 ALDH1A1 (1.00) CYP1A2CYP3A4TDP1ALDH1A1SLC6A4
SCHEMBL207554 0.67 ALDH1A1 (0.62) CYP1A2CYP3A4TDP1ALDH1A1SLC6A4
SCHEMBL29374052 0.67 ALDH1A1 (0.62) CYP1A2CYP3A4TDP1ALDH1A1SLC6A4
1-Naphthylisothiocyanate SCHEMBL27487887 0.67 ALDH1A1 (0.96) CYP1A2CYP3A4TDP1ALDH1A1SLC6A4
1-Naphthylisothiocyanate SCHEMBL27570428 0.67 ALDH1A1 (0.96) CYP1A2CYP3A4TDP1ALDH1A1SLC6A4
SCHEMBL98105 0.67 MEN1 (0.38) CYP1A2CYP3A4TDP1SLC6A4MAOA
SCHEMBL330963 0.66 ALDH1A1 (0.56) CYP1A2CYP3A4TDP1ALDH1A1SLC6A4
SCHEMBL1997655 0.66 ALDH1A1 (0.75) CYP1A2CYP3A4TDP1ALDH1A1SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4398028-A HYPOTENSIVE, MUSCLE RELAXANTS SANDOZ LTD. (CH) 1983-08-09 US disclosed
US-4297490-A HYPOTENSIVE AND ANTISPASMODIC AGENTS SANDOZ LTD. (CH) 1981-10-27 US disclosed